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[(2S,6S)-11-methoxy-4-[4-(trifluoromethyl)pyridin-2-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
methyl (1R,3S,3aR,6aS)-3-(dimethyl-1,2-oxazol-4-yl)-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-3-(pyridin-3-yl)propan-1-one
6-methyl-5-{2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,5S)-N-butyl-1-[(4-hydroxyphenyl)methyl]-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
N-ethyl-4-methanesulfonyl-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
N-benzyl-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-sulfonamide
N-butyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N,5-dimethyl-1H-pyrazole-4-carboxamide
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
1'-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
5-{[2-(3-phenylpyrrolidin-1-yl)ethyl]carbamoyl}thiophene-2-carboxylic acid
1-ethyl-4,6-dimethyl-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
(2-methoxyethyl)[(4-methylphenyl)methyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-(ethylamino)-5-methyl-N-[3-(propan-2-yloxy)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-{[8-(2,3,6-trimethylquinoline-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-3,3,3-trifluoropropanamide
4-ethyl-2-methyl-5-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1,3-thiazole
2-methoxy-1-[1'-(2-phenylacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
8-[(3,5-dimethylphenyl)methyl]-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
3-(2-fluoro-3-methoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-[4-(cycloheptylamino)-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-[3-(2-{[(2,4-dimethoxyphenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
(2S,4R)-4-amino-1-{2-[cyclopentyl(methyl)amino]acetyl}-N-ethylpyrrolidine-2-carboxamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-({5-[2-(3-chloro-1H-1,2,4-triazol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
2-amino-N-benzyl-4-methyl-N-[(6-methylpyridin-2-yl)methyl]pyrimidine-5-carboxamide
2-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-N-[2-(4-chlorophenyl)ethyl]acetamide
2-[2-(furan-2-yl)phenyl]-1-(2-methanesulfonylethyl)-1H-imidazole
2-(4-fluorophenoxymethyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-butyl-2-(4-{[(2-hydroxyethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-cyclohexyl-N5-cyclopropyl-N3-methyl-N3-[2-(4-methylphenoxy)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-hydroxy-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}pyrazine-2-carboxamide
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-2-[methyl(phenyl)amino]ethan-1-one
N-ethyl-N-(oxan-4-ylmethyl)-2-(1H-pyrazol-1-yl)butanamide
1-[(2-chlorophenyl)methyl]-N-(1,4-dioxan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
8-{[5-(4-chlorophenyl)furan-2-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(4-fluorophenyl)methyl]-3-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)propanamide
1-(pyridin-2-ylmethyl)-4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazine
2-{[4-(1H-imidazol-1-yl)butanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-[2-(dimethylamino)ethyl]-8-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-{[3-(furan-2-yl)phenyl]methyl}-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(2-methyl-1,3-thiazol-4-yl)-1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
2,6-dihydroxy-N-(1-methanesulfonylpiperidin-4-yl)benzamide
2-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-4-yl]-5-fluoro-1H-1,3-benzodiazole
N-(pyridin-2-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[3-(pyridin-4-yl)propyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide