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1-(6-fluoro-4-methylquinazolin-2-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}piperidin-4-amine
N-({7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,6-difluorobenzamide
N-({3-methyl-7-[(2E)-4-methylpent-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
1-[(2,4-difluorophenyl)methyl]-5-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}azepan-2-one
N-cyclopropyl-3-{1-[(2,4-dimethoxy-3-methylphenyl)methyl]piperidin-3-yl}propanamide
6-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(2-methoxyethyl)-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-ethyl-2-methyl-6-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
N-[2-(1H-imidazol-2-yl)ethyl]-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(4aS,8aR)-1-(2-phenylethyl)-6-(3,3,3-trifluoropropyl)-decahydro-1,6-naphthyridin-2-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(1H-pyrazol-1-yl)acetamide
7-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,3-oxazole
N-benzyl[(quinolin-6-yl)amino]sulfonamide
(furan-2-ylmethyl)({[3-(3-methoxyphenyl)oxolan-3-yl]methyl})(prop-2-en-1-yl)amine
1-(cyclopropylmethyl)-N-ethyl-5-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]amine
N-(1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-4-yl)methanesulfonamide
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(5-methylfuran-2-yl)methyl]piperidine
1-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-(piperidin-1-yl)propan-2-ol
N-(butan-2-yl)-4-{4-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine-1-carboxamide
methyl 1-{[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-2-carboxylate
5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1-[1-(thiophen-2-yl)ethyl]-1H-imidazole
2-(methylamino)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidin-3-yl]acetamide
(1-{[methyl({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl})amino]methyl}cyclopropyl)methanol
4-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,5,7-trimethylquinoline
N-[3-(4-{[2-(4-methoxyphenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
N-cyclopropyl-1-[(1s,4s)-4-[2-(3-chlorophenyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)phenyl]-1H-pyrazol-4-yl}pyridine-3-carboxamide
N-[2-(2-methylpropanesulfonyl)ethyl]-1,2-oxazole-3-carboxamide
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)-3,5-dimethoxybenzamide
N-[2-(adamantan-1-yl)ethyl]-5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-2-(pyrrolidin-1-yl)pyridine
methyl({[3-(2-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-2-yl}ethoxy)phenyl]methyl})(quinolin-8-ylmethyl)amine
2,5-dichloro-N-{2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}benzamide
5-(4-fluorophenyl)-4-[1-(1H-imidazole-4-carbonyl)piperidin-3-yl]-2-methylpyrimidine
4-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2,3-dimethoxybenzamide
[(3R,4R)-1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}azepan-2-one
5-[3-(3-benzoylpiperidin-1-yl)-3-oxopropyl]-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
ethyl 1-ethyl-5-{imidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]cyclopentanecarboxamide
4-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1H-imidazol-1-yl}benzene-1-sulfonamide
1-[(1-methylpiperidin-3-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-[2-(azepan-1-yl)ethyl]-N-ethyl-6-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide