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6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-propylpyridine-3-carboxamide
N3-ethyl-N5-(naphthalen-1-ylmethyl)-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[3-methyl-7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}methanesulfonamide
5-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-({[(3R,4R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-ethyl-1-[4-(furan-2-yl)benzoyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
4-{6-[1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-2-oxopentanamide
N-(2-{[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}ethyl)acetamide
2,4-dimethyl-N-[3-(morpholin-4-yl)propyl]-1,3-oxazole-5-carboxamide
3-(6-methoxynaphthalene-2-carbonyl)-1-(5-methyl-1H-pyrazole-3-carbonyl)piperidine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carboxamide
1-[(3-chlorophenyl)methyl]-3-(1H-imidazol-1-ylmethyl)piperidine
(2S)-2-{4-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}-3-(pyridin-4-yl)propanoic acid
1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
4-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(1r,4r)-4-{[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}cyclohexan-1-ol
(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)(pyridin-3-yl)methanol
N-[3-(propan-2-yloxy)propyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-tert-butyl-3-[(3E)-hex-3-enamido]-2-methylbenzamide
ethyl 3,5-dimethyl-4-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]-1H-pyrrole-2-carboxylate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-fluoro-2-methylbenzoyl)piperidin-3-ol
dimethyl({[5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)furan-2-yl]methyl})amine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-8-fluoroquinoline-2-carboxamide
1-(2-methoxyphenyl)-4-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperazin-2-one
(propan-2-yl)({[6-(trifluoromethyl)pyridin-3-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
ethyl 4-[(4-methoxyphenyl)methyl]-1-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetyl)piperidine-4-carboxylate
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2,5-dimethyl-N-(oxolan-2-ylmethyl)furan-3-carboxamide
(4aS,8aS)-2-cyclohexyl-7-(3-hydroxy-1,2-oxazole-5-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
2-[3-(pyrimidin-5-yl)phenoxy]propanamide
2-amino-6-(2-methylpropanoyl)-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(1S,5R)-3-(1-benzyl-1H-pyrazole-4-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl({4-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]phenyl}methyl)amine
5-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-cyclopentanecarbonyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
N-(propan-2-yl)-1-[(1s,4s)-4-[2-(4-methoxyphenoxy)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)[(5-methylthiophen-2-yl)methyl]amine
3-(1-ethyl-1H-imidazol-2-yl)-1-(3-fluoro-4-methoxybenzoyl)piperidine
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(3-methylthiophen-2-yl)methyl]amine
methyl 1-{3-[(4-methoxyphenyl)methyl]-1,2-oxazole-5-carbonyl}piperidine-2-carboxylate
(1R,5R)-3-benzoyl-6-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[1-(2-fluorophenyl)-1H-pyrazol-3-yl]-4-methyl-1,3-thiazol-2-amine
3-(1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidin-3-yl)propan-1-ol
2-[5-(5-chlorothiophen-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
8-[(4-ethylphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione