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N-(2,4-difluorophenyl)-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]morpholine-4-carboxamide
(1S,5R)-3-[2-(difluoromethoxy)benzoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-cyclopentylpiperidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-ethyl-N,2-dimethyl-N-[2-(piperidin-1-yl)ethyl]quinoline-4-carboxamide
1-methyl-4-({1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrazole
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-7-fluoro-N,2-dimethylquinoline-4-carboxamide
3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-(difluoromethyl)-1H-pyrazole
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
2-(2-hydroxyethyl)-6-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(oxolan-2-ylmethyl)piperazine
N-[4-(methylsulfanyl)phenyl]-6-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-dimethyl-5-[1-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
[5-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)furan-2-yl]methanol
[1-(thiophen-2-yl)ethyl][(5,6,7-trimethoxy-2-phenylquinolin-3-yl)methyl]amine
2,4-difluoro-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
methyl 5-[(1-acetylpiperidin-4-yl)amino]-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3aR,5R,6S,7aS)-2-[1-(4-phenoxyphenyl)-1H-1,2,3,4-tetrazol-5-yl]-octahydro-1H-isoindole-5,6-diol
1-[(1,5-dimethyl-1H-indol-2-yl)methyl]-N,N-dimethylpiperidin-3-amine
{5-[2-(2-ethylpyrimidin-4-yl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-2-yl}methanol
3-[2-(dimethylamino)ethyl]-5-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-butyl-4-(2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-1H-1,2,3-triazol-1-yl}propane-1,2-diol
5-[(1,3-benzothiazol-2-ylmethyl)amino]-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(3-methylthiophen-2-yl)methyl]-decahydro-2,7-naphthyridine-2-sulfonamide
methyl 2-(2-{[3-(furan-2-yl)propanamido]methyl}-5-methyl-2,3-dihydro-1-benzofuran-7-yl)benzoate
N-methyl-2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
5-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
1-cyclohexyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidine-4-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}propanamide
2,4-dichloro-3-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)phenol
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(3-hydroxyquinoxalin-2-yl)-N-methylpropanamide
1-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{2-[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4-methylpiperazine
2-tert-butyl-6-(4-ethoxy-3-methoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-benzyl-4-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-(3-fluoro-4-methoxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
N-[2-(2-chlorophenyl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
N-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-cyclopropyl-6-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1,3-benzoxazole
4-methoxy-N-(2-methoxyethyl)-2-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide