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N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-4-carbonitrile
1-(3-{[(2-hydroxyethyl)(methyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
[(3R,4R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
5-(2-methoxyphenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(1-methyl-1H-indazol-6-yl)urea
2-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]pyridine-4-carbonitrile
5-cyclopropyl-N-ethyl-N-(2-hydroxyethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(3aS,6aS)-2-[2-(pyridin-2-yl)acetyl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(oxolane-3-carbonyl)-1,4-diazepan-2-one
9-(2,3-dimethylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(4-fluorophenyl)-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-oxo-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
6-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine-2,4-diamine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(2-methylprop-2-en-1-yl)azepan-4-amine
2-({1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)morpholine
5-chloro-7-methoxy-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-benzofuran-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(2-methylpropyl)amino]methyl}piperidin-2-one
8-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(1S,5R)-3-cyclobutanecarbonyl-6-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(cyclopropylmethyl)-5-[(4-methoxyphenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3R,9aR)-8-(4-fluorobenzoyl)-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(4-cyano-4-methylpiperidine-1-carbonyl)-N-[(3R)-pyrrolidin-3-yl]benzene-1-sulfonamide
1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
5-{imidazo[1,2-a]pyridin-2-yl}-3-(2-methoxyphenyl)-1,2,4-oxadiazole
1-cycloheptyl-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-oxopiperidine-3-carboxamide
3-(4-hydroxyphenyl)-N-[(1-phenylcyclopentyl)methyl]-1H-pyrazole-5-carboxamide
2-butyl-8-[(2,3-dimethoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 1-({4-[2-(2-methoxyphenoxy)acetyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-2-carboxylate
2-(1H-pyrazol-1-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]butanamide
6-ethoxy-3-{[methyl(oxolan-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(1-cyclobutanecarbonylpiperidin-4-yl)-5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
1-(2-{[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)piperidin-3-ol
5-{1-[2-(morpholin-4-yl)propanoyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-3-(2-oxopyrrolidin-1-yl)benzamide
1-[(2-methoxyphenyl)methyl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(2,2-dimethyloxan-4-yl)pyrimidin-2-amine
methyl 1-{2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-4-carboxylate
2-(1H-indazol-1-yl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
1-[3-(furan-2-yl)benzoyl]-3-(2-methoxyphenoxy)azetidine
1-(cyclopropylmethyl)-5-[(2,4-dimethoxyphenyl)methyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-fluoro-5-sulfamoyl-N-(thiolan-3-yl)benzamide
3-methyl-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one