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2-benzyl-9-(2-hydroxypyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-chloro-N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
3,4,5-trimethoxy-N-[2-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)propyl]benzamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-{2-[2-(pentan-3-yl)-1H-imidazol-1-yl]ethyl}piperidine-3-carboxamide
N-({7-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
1-(diethylamino)-3-[4-({[(2-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
(4S)-1-[4-(4-fluorophenyl)benzoyl]-3,3,4-trimethylpiperidin-4-ol
1-[(1R,5R)-6-[(4-fluoro-3-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-phenyl-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine-4-carbonitrile
5-{1-[3-(2-chlorophenyl)propanoyl]piperidin-4-yl}-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
6-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyrimidin-4-amine
N-[4-(2-fluorophenoxy)phenyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-{3-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
(1R,3S)-3-(2-aminoethoxy)-7-[(2-cyclohexylpyrimidin-5-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
1-(5,6-dimethylpyrimidin-4-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
2-{5-[3-methyl-4-(morpholin-4-yl)phenyl]-3-(3-methylbutyl)-1H-1,2,4-triazol-1-yl}acetic acid
1-[(3-methylquinoxalin-2-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
1-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
N-methyl-2-(morpholin-4-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-(pyridin-3-yl)acetamide
(2E)-3-(3-fluorophenyl)-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
1-(benzyloxy)-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1,8-diazaspiro[4.5]decan-2-one
1-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)-4-phenylbutan-1-one
(4aS,8aR)-1-(2-aminoethyl)-6-[(4-methylthiophen-2-yl)sulfonyl]-decahydro-1,6-naphthyridin-2-one
N-(cyclopropylmethyl)-2-(4-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}[2-(1H-indol-3-yl)ethyl]amine
7-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[2-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(4-fluorophenoxy)piperidine
5-(cyclohex-3-ene-1-carbonyl)-3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
ethyl 1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
1-[1-(carbamoylmethyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
1-(cyclohexylmethyl)-N-(1-hydroxypropan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-[3-(4-fluorophenyl)propanoyl]-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
3-(2-amino-1,3-thiazol-4-yl)-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
2-chloro-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)pyridine-4-carboxamide
N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-3-(piperidin-3-yl)benzamide
3-[(3R,4S)-1-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-(3-chloro-5-methylpyridin-2-yl)-4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazine
ethyl 3-benzyl-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine-3-carboxylate
N-methyl-N-(2-phenoxyethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
N-{[7-(pyrimidin-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}but-3-enamide
2-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)-3-methoxyphenol
3-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}phenol
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-{imidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide