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5-(3-methylbut-2-en-1-yl)-1'-(pyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
1-(4-benzylpiperazin-1-yl)-3-[1-(furan-2-ylmethyl)piperidin-3-yl]propan-1-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
6-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]quinoxaline
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
3-[({[2-(butan-2-yl)phenyl]carbamoyl}amino)methyl]-N,N-dimethylbenzamide
1-(4-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}phenyl)imidazolidin-2-one
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
6-cyclopentyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-ethyl-5-oxopyrrolidine-3-carboxamide
1-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidine-4-carboxamide
(1S,3R)-N-(6-methoxypyridin-3-yl)-3-[2-(pyridin-4-yl)acetamido]cyclopentane-1-carboxamide
N-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-amine
methyl 5-{[(3-methylphenyl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-amino-N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)cyclopentane-1-carboxamide
N-[2-(2-ethoxyphenyl)ethyl]-2-methylpyrimidine-5-carboxamide
N-[3-(3-cyano-1H-pyrazol-4-yl)phenyl]acetamide
N,N-dimethyl-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-amine
N-(1-benzylpiperidin-3-yl)-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
5-(naphthalen-1-ylmethyl)-5-{3-oxo-3-[3-(pyridine-3-carbonyl)piperidin-1-yl]propyl}pyrrolidin-2-one
{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}(1-methoxypropan-2-yl)amine
7-fluoro-2-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-6-methyl-2,3-dihydropyridazin-3-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
1-{[(2R,5S)-5-(pyridin-3-ylmethyl)oxolan-2-yl]methyl}piperidine-4-carboxylic acid
7-(1,3-benzothiazol-2-yl)-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethan-1-one
4-(2-methyl-1H-imidazol-1-yl)-1-(thiophen-3-ylmethyl)piperidine-4-carboxylic acid
3,6-dimethyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(3-phenylpropyl)piperidin-4-ol
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(3,6-dimethylpyrazin-2-yl)piperidine-4-carboxylic acid
5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-[2-(piperidin-1-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-1-[(5-methylpyrazin-2-yl)methyl]urea
(3S,4R)-1-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(6-methylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[4-(2-chloro-6-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenol
3-chloro-N-(2-methoxyethyl)-4-({1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}oxy)benzamide
2-[4-({3-[(diethylamino)methyl]-4-methoxyphenyl}methyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
5,6-dimethyl-2-[4-(pyrimidin-5-yl)phenyl]-1H-1,3-benzodiazole
5-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]-2-(pyridin-2-yl)pyrimidine
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methoxypyrimidine
3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N-methylbenzamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-(quinazolin-4-yloxy)ethan-1-one
2-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-6-methoxyphenol
(3S,4R)-N,N-dimethyl-1-(4-methylquinolin-2-yl)-4-propylpyrrolidin-3-amine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[1-(pyridin-2-yl)propan-2-yl]piperazine
N-(2H-1,3-benzodioxol-5-yl)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-amine
2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(pyrrolidin-1-yl)pyrazine