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1-[2-(dimethylamino)-6-[(2S)-pyrrolidine-2-carbonyl]-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
4-(2-methoxyethyl)-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
5-(3-methoxyphenoxymethyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
4-[(4-methoxy-3-methylphenyl)methyl]-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]piperazin-2-one
5-(2-ethoxyphenyl)-N-ethylthiophene-2-carboxamide
(2R,6R)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[8-(2,3-dihydro-1H-indene-1-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]propanoic acid
1-{2-[2-(4-fluorophenyl)morpholin-4-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
4-methyl-2-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(thiophene-2-carbonyl)piperidin-3-amine
5-{1-[3-(4-methoxyphenyl)propanoyl]piperidin-4-yl}-5-(2-methylpropyl)-3-(thiophen-2-ylmethyl)imidazolidine-2,4-dione
N-cyclopropyl-3-acetamido-N-[(2-methoxyphenyl)methyl]benzamide
2-phenyl-N-{[7-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-[2-(methylsulfanyl)phenyl]-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]acetic acid
N-cyclohexyl-4-[2-(2-methyl-1,3-thiazol-4-yl)acetamido]piperidine-1-carboxamide
5-{[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]methyl}-N-ethylpyrimidin-2-amine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-phenylcyclopropyl)acetamide
N-(5-methanesulfonyl-2-methylphenyl)-4-(pyridin-4-yl)piperidine-1-carboxamide
4-amino-1-[2-(3-chlorophenyl)ethyl]pyrrolidin-2-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-ethyl-1,2-oxazole-5-carboxamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
(1R,5S)-8-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-3,8-diazabicyclo[3.2.1]octane
(2E)-N-({7-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
N-[2-(ethanesulfonyl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(3-hydroxyphenyl)methyl]piperidine-4-carboxylic acid
N-tert-butyl-1-(3-methylbutyl)-4-oxo-5-{4-[1-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
(3S,4R)-4-(hydroxymethyl)-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
(3aR,5R,6S,7aS)-2-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-octahydro-1H-isoindole-5,6-diol
N-[(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2,5-dimethylfuran-3-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(morpholine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-butyl-8-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
1-ethyl-5-(2-{[(4-fluorophenyl)methyl]sulfanyl}ethyl)-1H-1,2,4-triazole
2-chloro-4-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}phenol
N-[(3-methoxyphenyl)methyl]-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]propanamide
2-(phenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide
(5S,9aS,9bS)-5-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[2-(dimethylamino)ethyl]-8-(4-methyl-1H-imidazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclobutyl-2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-{2-[methyl(phenyl)amino]propyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
4-(5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
3-(5-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-[2-(methylsulfamoyl)ethyl]-2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine-3-carboxamide
(3S,4R)-1-[2-(2-ethoxyphenyl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine-2-carboxylic acid
4-(1H-1,3-benzodiazol-1-yl)-1-(2-methylpyridin-4-yl)piperidine-4-carboxylic acid
[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl](4-phenylbutan-2-yl)amine
1-(3-chlorophenyl)-4-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}piperazin-2-one
(3aS,6aS)-2-methyl-5-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid