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4-ethyl-3-{1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-[5-(methoxymethyl)furan-2-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-1λ6-thiomorpholine-1,1-dione
1-(4-chloro-2-hydroxybenzoyl)-3-[(dimethylamino)methyl]piperidin-3-ol
2-ethoxy-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(2S)-1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-hydroxy-3-phenylpropan-1-one
3-(5-{[5-(4-methylphenyl)furan-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
[(3R,4R)-1-benzoyl-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
N-[(2-chloropyridin-3-yl)methyl]-6-ethyl-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
(2S,4S)-4-amino-1-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 1-(1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)piperidine-2-carboxylate
5-methyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
2-(3,5-dimethoxyphenyl)-3-(pyrrolidin-1-yl)pyrazine
2-(4-{[4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazin-1-yl]methyl}phenoxy)acetic acid
5-cyclopentyl-3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
N-(2-{7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecan-3-yl}-2-oxoethyl)benzamide
3-{1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-2-yl}propanoic acid
N-(1-{[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
3-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
2-(2-chloro-6-fluorophenyl)-1-[2-(1H-imidazol-2-yl)ethyl]-1H-imidazole
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
4-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-1-(2-methylpropyl)pyrrolidin-2-one
N-[(3,5-dimethoxyphenyl)methyl]-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3R,4R)-4-methyl-3-(propan-2-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-3-ol
N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)quinoline-2-carboxamide
3-(3-acetylphenyl)-1-methyl-6-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
4-[(2,3-difluorophenyl)methyl]-3-{2-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
3-(5-methylfuran-2-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
(1R,2S,3S,4R,5S)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)tricyclo[3.2.1.02,4]octane-3-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(2-chlorophenoxy)azetidine
(4aS,7aR)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-[(pentan-3-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]-N-(2,2,2-trifluoroethyl)benzamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(propan-2-yloxy)benzamide
7-fluoro-3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)imidazolidine-2,4-dione
6-[2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-1H-indazole
3-ethyl-8-[3-(1H-imidazol-2-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-[(3-methylphenyl)methyl]-2-(5-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decane
(3S)-1-ethyl-3-methyl-4-{4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanoyl}piperazin-2-one
N-[3-(dimethylamino)phenyl]-3-{[(4-methyl-1H-imidazol-5-yl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one