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(1S,5R)-3-cyclopentanecarbonyl-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(cyclopentylamino)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-methylpentanamide
2-methyl-6-({[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amino}methyl)phenol
N-(1-{7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
1,4-dimethyl 2-({1-[4-(5-phenylpentanamido)phenyl]piperidin-4-yl}amino)butanedioate
3-(2H-1,3-benzodioxol-5-yl)-5-(2-methylpropyl)-1H-1,2,4-triazole
N-[2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-ol
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)acetamide
2-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(2,3-dihydro-1H-isoindol-2-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-[1-(5-fluoropyridine-2-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
N-cyclohexyl-N-[(3-methylphenyl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-(3-phenylpiperazin-1-yl)-5,6,7,8-tetrahydroquinazolin-2-amine
1-{4-[(propan-2-yloxy)methyl]piperidin-1-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
5-{[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-N-methylfuran-2-carboxamide
N-[(5,6-dimethylpyridin-3-yl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-cyclohexyl-2-(1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)butanamide
{[3-(4-ethylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
[(1-cyclopentylpiperidin-4-yl)methyl]({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
5-{2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-1H-1,2,3,4-tetrazole
1-methyl-3-[5-(3-oxo-3-phenylpropyl)-1,3,4-thiadiazol-2-yl]-1-(pyridin-2-ylmethyl)urea
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-{3-[(diethylamino)methyl]phenyl}-6-(4-fluorophenyl)-3,4-dihydropyrimidin-4-one
N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
3-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]-3-(4-methoxyphenyl)-1-(3-methylbutyl)pyrrolidine-2,5-dione
4-[4-(3-methylphenoxy)piperidin-1-yl]-4-oxobutane-1-sulfonamide
2-[cyclopentyl(methyl)amino]-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N,N-dimethyl-2-[(1S,5R)-3-[(5-methylfuran-2-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-4-(oxolane-2-carbonyl)-1,4-diazepane
N-methyl-4-(4-methylphenoxy)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)piperidine-4-carboxamide
3-[({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)methyl]pyridin-2-amine
1-(butan-2-yl)-N3-[(4-chlorophenyl)methyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-fluorophenoxymethyl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1,3-oxazole-4-carboxamide
(3S,5R)-1-[3-(methylsulfanyl)propyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-[(3S,4S)-3-hydroxy-4-[4-(2-methylphenoxy)piperidin-1-yl]pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-benzyl-2-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
6-methoxy-3-[3-(1H-pyrazol-3-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
1-cyclobutanecarbonyl-N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]piperidine-4-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
(3aS,6aS)-2-[(2,4-difluorophenyl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-(pyridine-3-carbonyl)-6-azaspiro[2.5]octane
N-ethyl-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
5-methanesulfonyl-2-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-4-(piperidin-3-yl)pyrimidine
3-[1-(oxolane-2-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-[(2-chloro-6-fluorophenyl)methyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
N-[1-(thian-4-yl)piperidin-4-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide