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N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[2-(2-methoxy-5-{[methyl(propan-2-yl)amino]methyl}phenoxy)propyl]naphthalene-1-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(5-methylthiophen-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-(2-aminoethyl)-6-(4-phenoxybutanoyl)-decahydro-1,6-naphthyridin-2-one
2-ethoxy-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
(4aR,7aS)-1-acetyl-4-[(4-phenoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,5-dimethyl-3-{4-[3-(piperidin-3-yl)benzoyl]piperazin-1-yl}pyrazine
4-({1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}amino)pyrimidine-5-carboxylic acid
5-methyl-5-{1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]piperidin-4-yl}-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-{1-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}pyridine-2-carboxamide
N-[1-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
3-methyl-7-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
8-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-(6-fluoro-4-methylquinazolin-2-yl)-N-methyl-N-(quinolin-5-ylmethyl)piperidine-4-carboxamide
3-(diethylamino)-N-(2,4,6-trimethylphenyl)pyrrolidine-1-carboxamide
(2R,3R)-3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(4-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}piperazin-1-yl)pyridine-3-carboxamide
N-[(3S,4R)-1-[(3-cyanophenyl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
N-(1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)acetamide
2,5-dimethyl-N-{3-[5-methyl-4-({[4-(propan-2-yloxy)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}furan-3-carboxamide
4-(piperidin-1-yl)-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]benzamide
2-[2-(3-cyanophenyl)phenoxy]propanamide
(1R,5S,6R)-3-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-cyclohexyl-6-(methoxymethyl)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
(1S,5R)-3-{[3-(methylsulfanyl)phenyl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
3-({[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
{1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
1-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
2-{[4-(2-chlorophenyl)-5-[(2-fluorophenyl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-(2,4-dimethylpyrimidine-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
4-chloro-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-3-methyl-1H-pyrazole-5-carboxamide
N-[(2-fluorophenyl)methyl]-5-(4-formylpiperazin-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
4-(2-methoxyphenoxy)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
N-[(2-chloro-6-fluorophenyl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-(4-chlorophenyl)-N-({1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(1-methoxybutan-2-yl)-1H-pyrazole-4-carboxamide
1,4-dimethyl-9-(2,6,8-trimethylquinoline-4-carbonyl)-1,4,9-triazaspiro[5.5]undecane
(2R,3S,6R)-5-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[4-(3-methoxypropyl)piperazine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
1-(2-chloroprop-2-en-1-yl)-3-{[(2-hydroxypropyl)amino]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
N-{3-[5-methyl-4-({[2-(methylsulfanyl)-1,3-thiazol-4-yl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}pyridine-2-carboxamide
2-amino-6-cyclopentyl-5-methyl-4-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]pyridine-3-carbonitrile
methyl 1-(2-methoxyethyl)-3-(2-phenylacetamido)-5-[(1-propylpiperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(5-methoxy-1H-indol-2-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
2-(5-fluoro-2-methylphenyl)benzamide
1-cyclopentyl-3-(2-fluorophenyl)-3-{2-oxo-2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]ethyl}pyrrolidine-2,5-dione
3-{[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(1H-imidazol-2-ylmethyl)piperidine