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2-[2,6-dimethyl-4-(piperidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
1-(furan-2-ylmethyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}piperidine-4-carboxamide
N-(2,4-dimethoxyphenyl)-3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propanamide
2,4-dimethyl-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}pyrimidine-5-carboxamide
N-(2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}ethyl)-2-chlorobenzamide
ethyl 1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
8-methoxy-N-methyl-N-[3-(morpholin-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-amine
[(3R,4R)-4-[(dimethylamino)methyl]-1-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}pyrrolidin-3-yl]methanol
4-[4-(4-ethylphenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N4-methyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine-2,4-diamine
(1S,5R)-3-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2R,6S)-2,6-dimethyl-4-{5-[(4-methylpiperazin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}morpholine
5-[methyl(2-phenylethyl)amino]-2-[3-(pyridin-3-yl)propyl]-2,3-dihydropyridazin-3-one
3-(3,4-dimethoxybenzoyl)-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
4-(5-methylpyridin-2-yl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-ol
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-4-methoxy-N-(pyridin-4-ylmethyl)benzamide
N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}but-3-enamide
{3-[(4-fluorophenyl)methyl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl}methanol
1-(furan-3-ylmethyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-cyclopropyl-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
5-({[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]amino}methyl)-N-methylfuran-2-carboxamide
2,4-dimethyl-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepane
2-{[(4-fluorophenyl)methyl](methyl)amino}-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2,3-dimethylpyridine
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]acetamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-indole
3-(4-chlorophenyl)-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)propan-1-ol
8-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[2-(1-cyclopentylpiperidin-4-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-(propan-2-yl)-4-(1,3-thiazole-5-carbonyl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
(2S,4R)-4-[(3-cyano-2-methoxypyridin-4-yl)amino]-N-methyl-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-3-[3-(4-methylphenyl)propanoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-(4H-1,2,4-triazol-4-yl)propanamide
1-(azocan-1-yl)-3-(2-methoxy-5-{[(2-methylpropyl)amino]methyl}phenoxy)propan-2-ol
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1-(pyrimidin-2-yl)piperidin-4-amine
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3-(hydroxymethyl)piperidin-3-ol
2-(3-fluorophenyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide
1-(carbamoylmethyl)-N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]piperidine-3-carboxamide
2-ethyl-4-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1,3-oxazole-5-carboxamide
3-(3-chlorophenyl)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}propan-1-one
methyl 1-[(3S,5S)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-(1-benzylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-[2-(4-fluoro-2-methylphenyl)acetyl]-1-methylpiperazine-2-carboxylic acid
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-N-{3-[(pyridin-3-yl)amino]propyl}-1-benzofuran-5-carboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol