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N-(2-methoxyethyl)-4-[3-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(methanesulfonylmethyl)-5-{[(2-methylphenyl)sulfanyl]methyl}-1,2,4-oxadiazole
2-(1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-2-yl)-6-methyl-1H-1,3-benzodiazole
1-(morpholin-4-yl)-3-{1-[2-(morpholin-4-yl)benzoyl]piperidin-3-yl}propan-1-one
(4aS,8aR)-1-butyl-6-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
ethyl 1-[1-(2-cycloheptyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]piperidine-4-carboxylate
N-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)methanesulfonamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
6-(3,5-difluoro-4-methoxybenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyridin-3-yl)piperidin-4-ol
5-{1-[2-(naphthalen-1-yl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-cyclohexyl-5-[2-(2-methyl-1H-imidazol-1-yl)propyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1'-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}spiro[indene-1,4'-piperidine]
(3aR,6aR)-2-acetyl-N-(furan-3-ylmethyl)-N-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[(1-phenylpyrrolidin-3-yl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-(3-methylpyridin-4-yl)-4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
2-(2-{1-[2-(5-acetylthiophen-3-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N,N-dimethyl-6-({[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}amino)pyridine-3-carboxamide
(3aR,6aS)-N-(2,6-dimethylphenyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(4-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[2-(3-{5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-2-oxoethyl]-2-sulfanylidene-1,3-thiazolidin-4-one
9-[3-(4-fluorophenyl)propanoyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
N-methyl-2-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-(thiophen-2-yl)acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-phenyl-N-{4-[4-({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}amino)piperidin-1-yl]phenyl}propanamide
1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
4-{1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}quinoline
2-amino-4-[3-(2-hydroxyethoxy)phenyl]-5-methyl-6-(propan-2-yl)pyridine-3-carbonitrile
2-(2,4-difluorophenoxy)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(1S)-1-phenylpropyl]amine
N-methyl-3-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}pyridin-2-amine
4-methyl-N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
3-(propan-2-yl)-5-[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[2-(dimethylamino)benzoyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[3-(morpholin-4-yl)azetidin-1-yl]ethan-1-one
N-(2-phenylethyl)-1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
3-(2,5-difluorobenzoyl)-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
N-[2-(azepan-1-yl)ethyl]-N-ethyl-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-ethyl-3-[(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-3-[5-(1,3-dihydroxypropan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
N-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{5-methoxy-2-[({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)methyl]phenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
methyl 2-{[5-acetamido-1-ethyl-2-(3-methoxyphenyl)-1H-1,3-benzodiazol-7-yl]formamido}acetate
(4aR,8aR)-4-(6-ethyl-2-methylquinoline-4-carbonyl)-octahydro-2H-1,4-benzoxazine
N-(1-cyclopentylpiperidin-4-yl)-3-(3-hydroxy-3-methylbutyl)benzamide
(3aS,6aS)-2-[(2-chlorophenyl)methyl]-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid