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1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(3-chlorophenyl)ethan-1-one
N-[6-methoxy-2-oxo-4-(1-phenyl-1H-pyrazol-5-yl)-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
({4-cyclopropyl-5-[1-(pyridine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5,7-dimethyl-N-(3-methyl-4-pentanamidophenyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(5-chloropyridin-2-yl)piperazine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-[2-(dimethylamino)ethyl]-N-methyl-5-oxo-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-3-carboxamide
6-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-methoxypyridine-4-carboxamide
N-{2-[(pyridin-3-yl)amino]ethyl}-4-(pyrrolidin-1-ylmethyl)benzamide
ethyl 1-(oxan-4-yl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-(dimethyl-1,2-oxazol-4-yl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
2-amino-6-(3,4-dimethoxyphenyl)-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
(1S,5R)-3-[4-(difluoromethoxy)benzoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(4-fluorophenyl)piperazin-2-one
methyl (2S,4R)-1-(1-ethylpiperidin-4-yl)-4-[3-(4-fluorophenyl)benzamido]pyrrolidine-2-carboxylate
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-[2-(propan-2-yloxy)ethyl]-1,4-dihydropyridine-3-carboxamide
1-(2-methoxyphenyl)-3-methyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1H-1,2,4-triazole-5-carboxamide
6-(1H-imidazol-1-yl)-9-methyl-2,3,4,9-tetrahydro-1H-carbazol-1-one
N-[(2R,3R)-2-methoxy-1'-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
2-methyl-6-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]pyrimidin-4-ol
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylquinoline-3-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
(1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(oxane-2-carbonyl)piperidine-4-carboxamide
1-(pyridin-2-ylmethyl)-5-(thiomorpholine-4-carbonyl)piperidin-2-one
4-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]-3,4-dihydrophthalazine-1-carboxamide
2-[(6-{pyrazolo[1,5-a]pyridin-7-yl}pyrazin-2-yl)sulfanyl]acetic acid
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-6-methylpyridine
N-[(2R,3R)-1'-(cyclopent-1-ene-1-carbonyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-(1H-1,2,4-triazol-3-yl)benzamide
methyl 1-{3-[4-({[3-(dimethylamino)-2,2-dimethylpropyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(thiophen-2-yl)propanamide
5-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-({1-[(6-ethoxyquinolin-2-yl)methyl]piperidin-3-yl}methyl)furan-2-carboxamide
(1R,2R,6S,7S)-4-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
methyl 2-{4-[(2,4-dimethylphenyl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-[2-(3-methoxypropyl)piperidin-1-yl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-cyclopentyl-4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
(3S,4R)-4-methyl-1-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)piperidine-3,4-diol
5-(2,2-difluorocyclopropanecarbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
methyl 3-(4-ethenylbenzoyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,5S)-3-(6-methyl-2-propylpyrimidin-4-yl)-3,8-diazabicyclo[3.2.1]octane
2-(2-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}phenoxy)acetic acid
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(2,4,5-trimethylbenzoyl)piperidine
N-[(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-2-carboxamide
1-{6-[3-(2-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyridin-3-yl}ethan-1-one
1-(5-phenyl-1,2-oxazole-4-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane