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methyl[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine
N,N-dimethyl-7-(naphthalene-1-sulfonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrazole-3-carbonyl)piperidine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-3-carboxamide
3-methyl-N-{1-[1-(2-oxo-4-phenylbutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
2-{4-[4-(3-methylphenoxy)piperidin-1-yl]piperidine-1-carbonyl}pyridine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
6-methyl-5-(3,4,5-trimethoxyphenyl)-1,3-benzothiazol-2-amine
4-methyl-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}pentane-1,2-dione
methyl({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-{4-[3-(methoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-methyl-5-{[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]quinoline-4-carboxamide
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-2-(4-propanoylphenoxy)acetamide
{4-[1-(2-methoxyphenyl)piperidin-4-yl]-1,4-oxazepan-6-yl}methanol
N-[2-(4-{[2-(2,3-difluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]cyclobutanecarboxamide
N-(adamantan-2-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
3-{2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamido}propanamide
6-ethyl-N2,N2-dimethyl-N4-[2-(oxolan-3-yl)ethyl]pyrimidine-2,4-diamine
[(2S,4R,5R)-5-(4-chlorophenyl)-4-{[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]methyl}-1-ethyl-2-methylpyrrolidin-2-yl]methanol
3-[(3R,4S)-1-[3-(3-chlorophenyl)propanoyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
4-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1-(4-methylphenyl)piperazin-2-one
4-(2-chlorophenoxy)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
3-{[4-methyl-6-({[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}amino)pyrimidin-2-yl]amino}phenol
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
2-{[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-1H-1,3-benzodiazole
3-(3-fluoro-4-methoxybenzoyl)-1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidine
4-[1-(2-methylbutyl)piperidin-3-yl]-5-phenyl-2-(pyridin-4-yl)pyrimidine
4-{2-[4-(hydroxymethyl)phenyl]acetyl}-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-(naphthalen-2-yloxy)-1-(1,4-oxazepan-4-yl)propan-1-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
2-[4-(1,3-oxazol-5-yl)benzoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
8-(4-fluorobenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(3,4-difluorophenyl)methyl]-8-[(2-oxo-1,3-oxazolidin-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-amino-N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4-methyl-1,3-benzothiazole-6-carboxamide
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-[3-(pyrazin-2-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(2-methoxyethyl)sulfamoyl]-5-(3-methyl-1H-pyrazol-1-yl)benzoic acid
3-{[ethyl(propan-2-yl)amino]methyl}-N-(pyridin-4-yl)benzamide
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-3-(1-methylpiperidin-2-yl)propanamide
4-{3-oxo-3-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]propyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-(1-ethyl-1H-1,2,4-triazol-5-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
7-chloro-N,3,5-trimethyl-N-(1,2-oxazol-3-ylmethyl)-1-benzofuran-2-carboxamide
2-benzyl-8-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
methyl (2S,3S)-2-(3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-3-methylpentanoate
(2S,4S)-4-amino-N-ethyl-1-({[(2-methylphenyl)methyl]carbamoyl}methyl)pyrrolidine-2-carboxamide
methyl 1-{3-[4-({[(4,6-dimethylpyrimidin-2-yl)methyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
1-ethyl-N-(3-methoxypropyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-[2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-(2-methoxyethyl)-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
3-({[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}methyl)-N-butyl-N-methylimidazo[1,2-a]pyridine-2-carboxamide