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(1S,5R)-6-[(4-ethoxy-3-methoxyphenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-(diphenylmethyl)-7-oxo-2-(pyridine-4-amido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
(2-{2-[1-(5-chloro-3-fluoropyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
3-ethyl-N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1-methyl-1H-pyrazole-5-carboxamide
1-[(4-fluoro-3-methoxyphenyl)methyl]-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
methyl 9-(benzyloxy)-3-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 4-[(3-fluorophenyl)methyl]-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidine-4-carboxylate
1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(methoxymethyl)piperidine
N-[(5-chloro-2-methoxyphenyl)methyl]-N,5-dimethyl-2-phenyl-1H-imidazole-4-carboxamide
N-[(2-methoxyphenyl)methyl]-2-{[(1R,2R,3R,5S)-2,6,6-trimethylbicyclo[3.1.1]heptan-3-yl]amino}acetamide
1-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propan-1-one
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(pyridin-3-ylmethyl)amine
1-(cyclopropylmethyl)-5-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(cyclohex-3-ene-1-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}-3-methoxyphenol
4-(1-{2-[ethyl(methyl)amino]acetyl}piperidin-3-yl)benzoic acid
methyl 8-[(2-chlorophenyl)methyl]-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-amino-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]-N-[1-(4-methylphenyl)ethyl]acetamide
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(3-phenylpropyl)acetamide
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2-methylphenyl)methyl]piperidine
(1R,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methanol
(4aS,7aR)-4-ethyl-N-(2-methoxy-5-methylphenyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[(3S,4R)-1-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1,3-dimethyl-6-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3-methyl-7-{2-[4-(methylsulfanyl)phenyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(piperidin-1-yl)acetamide
(2S)-3-phenyl-2-[2-(4-phenylpiperidin-1-yl)acetamido]propanamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]acetamide
(2R)-N1-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)pyrrolidine-1,2-dicarboxamide
N-methyl-1-{[2-(trifluoromethoxy)phenyl]methyl}piperidine-2-carboxamide
3-(4-chlorophenyl)-5-(2,3-dihydro-1-benzofuran-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(1R,2R,4R)-N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
N-[1-(1H-imidazol-2-ylmethyl)azepan-4-yl]-2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-(3-{[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]sulfonyl}-4-methoxyphenyl)acetic acid
(2S,4S)-4-amino-N-ethyl-1-(4-methoxy-2,3,6-trimethylbenzenesulfonyl)pyrrolidine-2-carboxamide
(1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methanol
[(3R,4R)-1-(1,3-benzothiazole-6-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-methylazepane-2-carboxamide
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-propoxypiperidine
8-[2-(1,2-benzoxazol-3-yl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-cyclopentyl-N,N-diethyl-4-oxo-5-(4-phenylazepane-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-methyl-4-[4-(piperidin-3-ylmethyl)benzoyl]piperazine
N-(4-chloro-3-methylphenyl)-2-{[2-methyl-1-(pyridin-2-yl)propyl]amino}acetamide
methyl N-{1-[({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)carbamoyl]ethyl}carbamate
N-[2-(3-methoxyphenyl)ethyl]-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
1-[(2-hydroxyphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide