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N-{2-[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}-4-methylbenzamide
2-hydroxy-N-[(3R,4S)-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N3-cyclopentyl-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{2-amino-6-[(4-methylphenyl)sulfanyl]pyrimidin-4-yl}-4-hydroxypiperidine-4-carboxylic acid
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-[(cycloheptylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-{3-cyclopentyl-5-[2-(dimethylamino)pyridin-3-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-{2-[2-(1-benzofuran-5-yl)-1H-imidazol-1-yl]ethyl}pyridine-4-carboxamide
6-cyclopropyl-2-(4-{[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-5-(2,3,6-trifluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{4-[(2,3-difluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-methoxy-N-methyl-3-(morpholin-4-yl)-N-[1-(pyridin-3-yl)ethyl]benzamide
1-(4-ethylpiperazin-1-yl)-3-[1-(5-hydroxypyrazine-2-carbonyl)piperidin-4-yl]propan-1-one
4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
N-(furan-2-ylmethyl)-4-(hydroxymethyl)-N-(3-methylbutan-2-yl)benzamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(pentan-3-yl)-2,7-diazaspiro[4.5]decan-6-one
benzyl (3R,9R)-2,8-dioxo-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-11-carboxylate
N-cyclopropyl-2-(4-methyl-1,4-diazepan-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
(1S,5R)-3-(pyrimidin-2-yl)-N-(thiophen-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-(1H-indol-4-ylmethyl)-6-(2-methoxyphenyl)pyridazin-3-amine
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}oxane-2-carboxamide
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carboxamide
4-[1-(2-phenylethyl)pyrrolidin-3-yl]-2-(pyridin-4-yl)pyridine
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
[4-(2-phenoxyethyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl]methanol
ethyl 1-[2-(3-chlorophenoxy)propanoyl]-4-(cyclopropylmethyl)piperidine-4-carboxylate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-chloro-N,1,5-trimethyl-1H-pyrazole-3-carboxamide
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[4-(trifluoromethoxy)phenyl]methyl}propanamide
4-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperazine-2-carboxylic acid
N-(2,4-dimethoxyphenyl)-N'-[2-(dimethylamino)-1-phenylethyl]-N'-methylpropanediamide
5-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)imidazolidine-2,4-dione
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-methyl-1,2-oxazole-5-carboxamide
1-[4-(morpholine-4-carbonyl)phenyl]-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]piperidin-4-amine
9-methoxy-N-methyl-7-oxo-3-(2-phenylpropanoyl)-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-chloro-6-{methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}pyridine-2-carboxylic acid
3,5-dimethyl-4-oxo-N-[1-(pyridin-3-yl)pentyl]-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-1-(6-methoxy-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
7-methoxy-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1-{1-[(4-methyl-2-phenylpyrimidin-5-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
1-{4-[(cyclopent-3-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
1-(2-methoxyethyl)-4-[4-(pyridin-4-yl)piperidine-1-carbonyl]pyrrolidin-2-one
4-(2,4-dioxoimidazolidin-1-yl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}benzamide
N-(1,4-oxazepan-6-ylmethyl)-2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
9-methoxy-3-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(3aS,6aS)-2-methyl-5-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[2-(azocan-1-yl)acetyl]-1-methylpiperazine-2-carboxylic acid
N,N-dimethyl-6-[4-(1H-pyrazol-5-yl)phenyl]pyridine-2-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
6-methoxy-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-methyl-1-benzofuran-2-carboxamide