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(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[(3,5-dimethylphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-2-methyl-2-phenylpropan-1-one
N-(adamantan-2-yl)-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
2-(2-methoxyphenoxy)-1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(2S,4S)-4-amino-N,N-diethyl-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine-2-carboxamide
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-cyclopropyl-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperazine-2-carboxamide
1-{[5-(1-cyclobutanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}-4-methylpiperazine
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
N-(3-chloro-4-fluorophenyl)-3-(1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
1-[(3-methoxyphenyl)methyl]-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[(2-chlorophenyl)methyl]-3-{1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-3-yl}propanamide
3-(3-methoxypropyl)-1-[2-(trifluoromethyl)benzoyl]piperidine-3-carboxylic acid
4-(4-chlorophenyl)-1-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]butan-1-one
3-(2-amino-1,3-thiazol-4-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]propan-1-one
(2R)-2-cyclohexyl-2-hydroxy-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(furan-2-ylmethyl)-5-{1-[2-(2-methyl-1H-indol-3-yl)acetyl]piperidin-4-yl}-5-propylimidazolidine-2,4-dione
4-(1-benzofuran-2-yl)-2-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
4-[({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}amino)methyl]-1-ethylpyrrolidin-2-one
methyl 1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazole-3-carboxylate
N-(1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
N-(1,3-benzothiazol-2-ylmethyl)-N,2,5-trimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}furan-2-carboxamide
(2S,4S)-4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(thian-4-yl)piperidine-3-carboxamide
(2S,4R)-N,N-diethyl-1-(furan-3-carbonyl)-4-(3-hydroxypropanamido)pyrrolidine-2-carboxamide
5-{[(2-amino-5-ethylpyrimidin-4-yl)amino]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
(3S,4S)-4-cyclopropyl-1-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]pyrrolidine-3-carboxylic acid
1-(oxan-4-yl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-(dimethylamino)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylbenzamide
2-(4-fluorophenyl)-1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidine
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-2-(propan-2-yl)pyrimidine-4-carboxamide
1-benzyl-3-(2-methylphenyl)-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}pyrrolidine-2,5-dione
(4aR,8aS)-6-[(2,6-difluorophenyl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
3-ethyl-2-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-1H-indole
2-(3-{[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}phenoxy)acetic acid
3-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
4-({4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-2-(pyridin-4-yl)acetamide
3-ethyl-5-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-oxazole-4-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]acetamide
N-({1-[(2-hydroxy-6-methoxyquinolin-3-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
7-[(3-methylpyridin-4-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-acetyl-8-[2-(2-chloro-4-fluorophenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-[2-(5-methylfuran-2-yl)ethyl]pyridin-2-amine
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-(morpholin-4-yl)propyl]propanamide
2-[(4aR,7aS)-4-[(5-cyano-1H-pyrrol-3-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-fluoro-2-methylphenyl)methyl]piperidine
1-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one