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2-[1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]urea
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-(1H-pyrrole-3-carbonyl)pyrrolidin-3-amine
(3R,4R)-1-(4-methoxybenzoyl)-4-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyrrolidin-3-ol
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-(2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
(2E)-1-[(4aR,8aR)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-6-yl]-2-methylbut-2-en-1-one
2-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
2-(4-{[7-(1-hydroxy-2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenoxy)ethan-1-ol
6-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
1-phenyl-4-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}piperazine
6-methyl-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)pyridine-2-carboxamide
1-[(4aR,8aR)-4a-hydroxy-7-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
7-[3-(2-hydroxyphenyl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)thiomorpholine
1-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}azetidin-3-ol
(4aS,8aR)-6-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidine-4-carboxamide
7-[3-(1,3-benzothiazol-2-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane
methyl 3-{1-[(3-phenyl-1,2,4-thiadiazol-5-yl)carbamoyl]piperidin-4-yl}propanoate
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-4-methyl-1,3-thiazole-5-carboxamide
1'-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}spiro[indene-1,4'-piperidine]
2-(2-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
6-(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
6-chloro-8-methyl-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
3-(4-methylphenyl)-3-phenyl-1-(pyrrolidin-1-yl)propan-1-one
4-(4-propyl-1H-1,2,3-triazol-1-yl)-1-(thiophene-2-sulfonyl)piperidine
6-(methoxymethyl)-1-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(morpholin-3-yl)ethan-1-one
6,7-dimethoxy-2-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1,2,3,4-tetrahydroisoquinoline
4-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[2-(2-hydroxyethyl)piperidin-1-yl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
methyl (2R)-2-(4-hydroxyphenyl)-2-{[2-(morpholin-4-yl)phenyl]formamido}acetate
5-ethyl-N4-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}pyrimidine-2,4-diamine
N-cyclopropyl-1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-(cyclopropylmethyl)-5-[2-(2H-indazol-2-yl)acetyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-ethyl-1-methyl-N-{[3-methyl-7-(4-methylbenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-pyrazole-5-carboxamide
4-ethyl-3-[(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(1,3-dimethyl-4-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
N-{3-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}acetamide
N-[(5-chlorothiophen-2-yl)methyl]-1-(4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(thiomorpholin-4-yl)pyridine-3-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
N-methyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-(oxolan-2-ylmethyl)-N-{[4-(pyridin-3-ylmethoxy)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide