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5-({[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-2-methoxybenzoic acid
4-ethyl-6-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methylpyrimidine
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{2-[3-(3-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}urea
{3-[(3-chlorophenyl)methyl]-1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-3-yl}methanol
3-(3-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)benzoic acid
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-{[8-(pyridin-3-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-(2,4,6-trifluorophenyl)acetamide
(3S,4S)-1-(1-benzofuran-2-ylmethyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
4-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)morpholine
N-(4-methoxyphenyl)-1-(pyridine-4-carbonyl)piperidin-3-amine
3-(4-methoxyphenyl)-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(3-hydroxy-2,2-dimethylpropyl)propanamide
2-(2-chloro-6-fluorobenzamido)-N-[(3,5-difluorophenyl)methyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
6-[6-hydroxy-4-(1H-indol-2-ylmethyl)-1,4-diazepan-1-yl]pyridine-2-carbonitrile
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(3,5-dichlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 4-(2-{[(2-fluorophenyl)formamido]methyl}-1-oxa-8-azaspiro[4.5]decane-8-carbonyl)benzoate
N-cyclohexyl-N-methyl-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]pyrimidin-2-amine
N-methyl-N-[4-(morpholin-4-yl)butyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
7-[(3,4-difluorophenyl)methyl]-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decane
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-{1-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-[3-(trifluoromethyl)benzoyl]piperidine
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridine-3-carbonitrile
5-(1-hydroxycyclopentanecarbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[3-(2-chloro-4-fluorophenyl)phenyl]ethan-1-amine
5-tert-butyl-4-({1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)furan-2-carboxamide
N-ethyl-3-methyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}but-2-enamide
N-(4-fluoro-2-methylphenyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridin-3-ylformamido}propanamide
2-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
4-(5-amino-1H-pyrazole-3-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
methyl 1-(benzyloxy)-8-[(2-methylphenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(2-oxopyrrolidin-1-yl)propanamide
2-{1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl}-N-methyl-N-(2-methylpropyl)acetamide
3-(3,4-dimethoxyphenyl)-N-(1-methoxypropan-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
5-fluoro-2-(1H-indol-5-yl)-N,N-dimethylpyrimidin-4-amine
(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)-N-methyl-N-(propan-2-yl)pyrrolidine-1-sulfonamide
N-cyclopentyl-2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}propanamide
(3S,5R)-N3-cyclopentyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]piperidine-3,5-dicarboxamide
2-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)pyridine-3-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
6-fluoro-2-[2-(morpholin-4-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-1,3-benzodiazole
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(morpholin-4-yl)-2-oxoacetyl]pyrrolidine-3-carboxylic acid
{4-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]-1,4-oxazepan-6-yl}methanol
(2E)-N-{[5-fluoro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
2-(2-chlorophenyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}acetamide
1-(2-methylpropyl)-8-[1-(methylsulfanyl)propan-2-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 1-methoxy-8-[(3-methylquinoxalin-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate