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N-(3,4-dimethylphenyl)-3-[2-(methylsulfanyl)benzoyl]piperidine-1-carboxamide
N3-methyl-4-oxo-1-(3-phenylpropyl)-N5-[(3,4,5-trifluorophenyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one
4-({1-[(2R)-2-aminopropanoyl]piperidin-4-yl}oxy)-N-(2-phenylethyl)benzamide
2-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]acetamide
3-(4-chlorobenzoyl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidine
5-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
7-[(4-benzylpiperazin-1-yl)methyl]-5-(2-chloroprop-2-en-1-yl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-methyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
4-(2-methyl-4-phenylpyridine-3-carbonyl)-2-(trifluoromethyl)morpholine
5-butyl-4-methyl-6-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}pyrimidin-2-amine
2-(3-fluorophenoxymethyl)-4-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1,3-oxazole
2-(3-methoxyphenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
3,5-dimethyl-4-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
N-(2-hydroxyethyl)-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-propylacetamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-(dimethyl-1H-1,2,4-triazol-1-yl)ethan-1-one
N-(furan-2-ylmethyl)-5-{1-[2-(4-methoxyphenyl)ethyl]-1H-pyrazol-3-yl}-4-methyl-1,3-thiazol-2-amine
N-ethyl-2-{4-[4-(4-methoxyphenyl)butanoyl]piperazin-1-yl}acetamide
2-(cyclopropylmethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
6-(2,3-dimethylquinoxaline-6-carbonyl)-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[1-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylbenzamide
methyl 2-oxo-8-{[4-(propan-2-yl)phenyl]methyl}-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)quinoxaline
2-({4-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)morpholine
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-2-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
2-(4-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-1-cyclohexylpiperazin-2-yl)ethan-1-ol
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
3-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
(1S,5R)-3-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-methoxypropan-1-one
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-5,6-dimethylpyrimidin-4-amine
8-chloro-2-ethyl-4-[(2,3,4-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-7-fluoro-1-[2-(phenylsulfanyl)ethyl]-1,2-dihydroquinolin-2-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-chloro-N-cyclopentyl-4-{[1-(thiolan-3-yl)piperidin-4-yl]oxy}benzamide
ethyl 1-[(3-{[1-(3-chlorobenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
2-ethyl-9-[(2-fluoro-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-1-{1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(3aS,6aS)-2-[(2,4-dimethylphenyl)methyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-tert-butylbenzamido)cyclopentane-1-carboxylic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}-1,4-diazepan-5-one
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-ol
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
4-(4-fluoro-3-methoxyphenyl)-7-hydroxy-2-oxo-1,2,3,4-tetrahydroquinoline-6-carboxylic acid