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4-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
N-({1-[(3-cyanophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-N-methylfuran-2-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]benzamide
ethyl 3-(2-methoxyethyl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidine-3-carboxylate
2-hydroxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}butan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-3-[2-(methylsulfanyl)ethyl]-5-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-1,2,4-triazole
(3R,4R)-1-[3-(4-fluorophenoxy)propyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-(9H-fluoren-9-yl)-1-[2-(3-methoxypropyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5,7-trimethyl-1H-indole-2-carboxamide
ethyl 1-benzyl-5-[2-(5-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine-3-carbonyl}pyridine
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[3-(2-methylphenoxymethyl)piperidin-1-yl]propan-1-one
4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(methylamino)-1,3-thiazole-5-carboxamide
4,5-dimethyl 1-[(3S,5S)-5-[(furan-2-ylmethyl)carbamoyl]-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
(3S,5S)-1-(1-benzofuran-2-ylmethyl)-5-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
2-[1-(cyclohexylmethyl)-4-(pyridin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
2-(2-fluorobenzenesulfonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-butyl-N-(furan-2-ylmethyl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
4-[3-(4-fluorophenoxy)propyl]-1,4-oxazepan-5-one
2-amino-6-phenyl-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-[2-butyl-4-(2-methoxyphenyl)-5-oxopiperazin-1-yl]-4-oxobutanamide
N-methyl-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
3-(3-fluorophenyl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
1-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}pyrrolidin-2-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(pyrimidin-4-ylmethyl)acetamide
2-chloro-6-methoxy-3-{1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenol
3-{2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-1H-indole
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[2-(pyridin-3-yl)ethyl]piperidine-4-carboxamide
3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-N-(trimethyl-1H-pyrazol-4-yl)benzamide
1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-4-ol
3-({2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyridin-2-amine
(2R)-2-amino-N,4-dimethyl-N-[(3-methylthiophen-2-yl)methyl]pentanamide
N-[3-(2-oxopyrrolidin-1-yl)propyl]-2,3-dihydro-1H-indene-1-carboxamide
4-(2-methyl-6-{1-[(2R)-pyrrolidine-2-carbonyl]piperidin-4-yl}pyrimidin-4-yl)morpholine
3-(methylsulfanyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
N-[4-({4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]acetamide
N-cyclohexyl-1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
3-{2-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
N,N-dimethyl-1-(5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-3-amine
(2R,6R)-4-[(dimethyl-1,2-oxazol-4-yl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-{[3-chloro-5-(trifluoromethyl)pyridin-2-yl]methyl}-1λ6-thiane-1,1-dione
N-cyclohexyl-N-methyl-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-methyl-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydroquinoline-3-carboxamide
2-[({5-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
(3S,4R)-1-(2-amino-2-methylpropanoyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-methyl-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
3-(azocan-1-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]propanamide
3-cyclopropyl-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide