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4-[5-(2-chloro-4-fluorophenyl)-3-(ethoxymethyl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
(2S)-2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-3-hydroxypropanamide
(1R,3S)-3-methoxy-3-methyl-7-(oxan-4-ylmethyl)-7-azaspiro[3.5]nonan-1-ol
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-(thiomorpholin-4-yl)ethan-1-one
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
2-methyl-6-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(3S,5S,9R)-5-({[4-(propan-2-yl)phenyl]methyl}amino)-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
N-cyclopropyl-2-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}benzamide
N-[2-(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclobutanecarboxamide
N-[3-({[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-(pyrimidin-4-ylmethyl)acetamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
3-(4-methyl-1,3-thiazol-5-yl)-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}propanamide
7-[3-(5-methylfuran-2-yl)benzoyl]-1-oxa-7-azaspiro[3.5]nonane
2-[4-(1H-indol-2-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
(1S,5R)-3-({7-chloro-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(3-chloro-1,2-oxazol-5-yl)propan-1-one
1-{[4-methyl-5-(1-methylpiperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
N-[2-(2-fluorophenyl)-1-{1-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]piperidin-4-yl}ethyl]-N,2-dimethylfuran-3-carboxamide
(3S)-3-ethyl-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]morpholine
2-(3-fluorophenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
8-(1H-indazol-5-yl)quinoline
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-2,3-dihydro-1-benzofuran-2-carboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
3-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
2-methoxy-N-[(2R,3R)-1'-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
N-[(3-methoxy-2-propoxyphenyl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
2-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-5-(methanesulfonylmethyl)pyridine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)propanamide
3-[4-(oxolan-2-yl)butyl]-1-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
2-(4-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
1-(4-{[1-(4-fluorophenyl)pyrrolidin-3-yl]amino}piperidin-1-yl)-3-methylbutan-1-one
N-{[8-(3,3-dimethylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
8-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
9-(1H-pyrrole-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-(5-methylpyridin-2-yl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidin-4-ol
(2R)-2-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)propanamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-{[(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
N-(oxan-4-ylmethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,7-diazaspiro[4.5]decane
7-fluoro-2-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)quinoline-4-carboxamide
3-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-4,7-dimethyl-2,3-dihydro-1H-indol-2-one
2-{2-[1-(quinoline-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
6-ethyl-2-{3-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]phenyl}-3,4-dihydropyrimidin-4-one
4-oxo-N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}-3,4-dihydroquinazoline-2-carboxamide