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3-methoxy-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
(3R,4S)-4-cyclopropyl-1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-amine
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(benzyloxy)-1-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
5-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
N-[1-(cyclohexylmethyl)piperidin-3-yl]-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1,4-dithiepan-6-amine
1-(but-3-enoyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
1-[(2-amino-5-ethylpyrimidin-4-yl)amino]-3-(4-methylphenoxy)propan-2-ol
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)cyclohexanecarboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[(2-methylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(3S,4R)-1-[4-methoxy-3-(morpholin-4-yl)benzoyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
N-ethyl-5-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrazine-2-carboxamide
1-[(4aR,8aR)-1-(5-phenoxyfuran-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(2-methoxyphenyl)ethan-1-one
N-({1-[(5-hydroxy-2-methoxyphenyl)methyl]piperidin-3-yl}methyl)cyclobutanecarboxamide
3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
5-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-N-methylfuran-2-carboxamide
2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-N-(thiophen-2-ylmethyl)acetamide
4-[1-(2-fluorobenzoyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
7-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-[({[4-(3-chlorophenyl)-5-[(3-hydroxypropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-6-ethoxyphenol
5-butyl-1'-(pyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
methyl 3-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl)benzoate
N-cyclohexyl-1-(6-methoxy-4-methylquinazolin-2-yl)piperidin-4-amine
N-ethyl-N-(2-methoxyethyl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
7-fluoro-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-3-methyl-1-benzofuran-2-carboxamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-ethylpyrrolidine-3-carboxamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-3-(2,5-dioxoimidazolidin-4-yl)propanamide
1-(2-cyclohexylethyl)-3-hydroxy-3-{[methyl(oxan-4-yl)amino]methyl}piperidin-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)acetamide
7-[2-(oxolan-3-yl)-1H-imidazol-1-yl]-2,3,4,9-tetrahydro-1H-carbazol-1-one
3-chloro-N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzamide
1-{4-[1-(prop-2-en-1-yl)-1H-imidazol-2-yl]phenyl}ethan-1-one
1-(5-ethylthiophene-3-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
(1R,5R)-6-[(3-methyl-1-benzofuran-2-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[(2S)-1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]methanol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(2,5-dimethylphenoxymethyl)-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1,2-oxazole-3-carboxamide
2-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
2-(benzyloxy)-1-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
[1-(3,5-difluorobenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
3-[(4-methoxyphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)propyl]-1,2-oxazole-5-carboxamide
N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
3-ethyl-4-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperazin-2-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-(4-methoxyphenyl)-N-methylpropanamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(propan-2-yloxy)propanamide
5-(2,6-difluorophenoxymethyl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1,2-oxazole-3-carboxamide
N-[3-(4-fluorophenyl)phenyl]-1-{[5-(hydroxymethyl)furan-2-yl]methyl}pyrrolidine-2-carboxamide