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methyl 4-{4-[(4-hydroxy-2-methoxyphenyl)methyl]piperazin-1-yl}benzoate
2-methyl-9-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(2-{[4-(oxolan-3-ylmethyl)piperazin-1-yl]methyl}phenyl)methanol
N-({7-[3-(3-methoxyphenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
N-methyl-N-[(3-methyloxetan-3-yl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-benzyl-6-(pyridin-2-ylmethoxy)-4-[4-(thiophen-2-yl)butanoyl]-1,4-diazepan-2-one
1-[2-(dimethylamino)-2,3-dihydro-1H-indene-2-carbonyl]-4-(pyridin-2-yl)piperidin-4-ol
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[4-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2,2-dimethylpropan-1-one
4-(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)thiomorpholine
1'-[2-(3-hydroxyphenyl)acetyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(3R,4R)-4-[(6-chloro-8-methylquinolin-4-yl)amino]piperidin-3-ol
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]propanamide
5-{[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]methyl}-N-methylfuran-2-carboxamide
(1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-3-(3-phenylpropyl)piperidin-3-yl)methanol
5-(5-methyl-1,2-oxazol-3-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(1-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
N,N-diethyl-1-({4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
2-(2-hydroxyethyl)-8-[4-(hydroxymethyl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
6,7-dimethyl-2-(3,3,3-trifluoropropyl)-1H-1,3-benzodiazole
N-({7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-fluorobenzamide
2-{4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carbonitrile
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
1-{2-[(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amino]pyrimidin-4-yl}piperidin-3-ol
N-(3-methoxyphenyl)-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}propanamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]propan-1-one
N-[(3,5-dimethoxyphenyl)methyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-3-carboxamide
N-(furan-2-ylmethyl)-9-methoxy-7-oxo-3-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
N-{2-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)morpholin-2-yl]ethyl}acetamide
2-(3-hydroxyphenyl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)acetamide
(1R,5R)-6-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-[(3S,4R)-1-(2-methoxy-4-methylbenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-cyclopropyl-1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperazine-2-carboxamide
N,N-diethyl-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]pyridin-2-amine
3-{2-[3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
N-{4-[4-(butylamino)piperidin-1-yl]phenyl}-4-methoxybenzamide
1-cyclopropyl-3-(4-methoxyphenyl)-3-[2-oxo-2-(piperidin-1-yl)ethyl]pyrrolidine-2,5-dione
3-(pyridin-4-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
methyl 1-({4-[4-(piperidin-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl})methylamine
(2E)-3-(3-fluorophenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
6-methyl-2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
4-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]-1-(2-methoxyphenyl)piperazin-2-one
4-[5-(furan-3-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]benzonitrile
N-methyl-N-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[({[5-(2-methoxyacetamido)-2-methylphenyl]carbamoyl}amino)methyl]-N,N-dimethylfuran-2-carboxamide