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(2S,4S)-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-methyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
4-[3-(1-methoxyethyl)phenyl]-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
6-[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-6-yl]pyridine-2-carbonitrile
(3R,4R)-4-cyclobutyl-4-hydroxy-N-(4-methoxyphenyl)-3-methylpiperidine-1-carboxamide
N-(2-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-methyl-5-(propan-2-yl)-N-(1,3-thiazol-4-ylmethyl)-1H-pyrazole-4-carboxamide
5-methyl-5-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{2-[(4-methoxyphenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)piperidine-3-carboxamide
N-methyl-5-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]furan-2-carboxamide
2-(1H-indol-4-yl)pyridine-4-carbonitrile
3-{[2-(3,4-difluorophenyl)-1H-imidazol-1-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(4-methoxy-3-methylphenyl)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
N-(2-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)-2-(trifluoromethyl)benzamide
N-(4-methoxyphenyl)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[3-cyclopentyl-1-(2,5-dichlorophenyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
(1R,5R)-6-methyl-N-(naphthalen-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-cyclopropyl-N-[2-(5-methylfuran-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(3-methoxyphenyl)-4-{3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperazin-2-one
3-(diphenylmethyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-5-carboxamide
4,4-difluoro-1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
(4S)-4-(propan-2-yl)-3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-oxazolidin-2-one
2,2-dimethyl-1-{4-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]piperazin-1-yl}propan-1-one
3-{[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
1-(2-methoxyphenyl)-2,2-dimethyl-4-(6-methylpyridine-3-carbonyl)piperazine
3-chloro-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-fluoro-N-methyl-1-benzothiophene-2-carboxamide
N-({2-[3-(2,5-dimethylfuran-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-ethyl-5-{4-phenyl-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-5-yl}-1H-1,2,4-triazole
5-[(1-methyl-1H-indol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
3-({4-[1-(2-methyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
N-[(3,5-difluorophenyl)methyl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
3-(propan-2-yl)-1-{[1-(quinolin-4-ylmethyl)piperidin-3-yl]methyl}urea
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-fluorophenyl)methyl]piperidine
2-{[(4-hydroxybutyl)amino]methyl}-6-methylquinolin-4-ol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
1-cyclohexyl-N3-[furan-2-yl(phenyl)methyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[3-(3-methoxypropyl)piperidine-1-carbonyl]-5-methylphenol
1-[cyclohexyl(methyl)amino]-3-(2-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
2-amino-N-[1-(4-fluorophenyl)piperidin-4-yl]-6-(propan-2-yl)pyrimidine-4-carboxamide
2-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyridine
4-[1,5-bis(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
4-{1-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperidin-3-yl}morpholine
4-(5-{[(2,6-dimethylpyridin-3-yl)oxy]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
2-(2-hydroxypropyl)-9-methanesulfonyl-2,9-diazaspiro[5.5]undecan-3-one
4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-methyl-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
[(1-ethylpiperidin-3-yl)methyl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
2-(2-methoxyphenyl)quinoline
ethyl 4-[(5S,9aS,9bS)-2-(3-methoxyphenyl)-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
N-[(2R,3R)-2-hydroxy-1'-[(2,3,6-trifluorophenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide