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1-{3-[(pentan-3-yl)amino]propyl}piperidin-3-ol
4-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]azetidin-3-yl}pyridine
4-(4-{[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(2S,4R)-4-amino-1-(1-benzyl-1H-pyrazole-4-carbonyl)-N-ethylpyrrolidine-2-carboxamide
2-[(4-{4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)methyl]pyridine
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
6-{[5-(2-chlorophenyl)furan-2-yl]methyl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol
N-(2-chlorophenyl)-3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]propanamide
1'-(2H-1,3-benzodioxol-5-ylmethyl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 2-[(5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidin-6-yl)formamido]acetate
N-({7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
3-[1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)piperidin-4-yl]benzonitrile
2-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[(2,4-dimethoxyphenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)pyridine
methyl (1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
1-[(2,4-difluorophenyl)methyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(cyclopropylmethyl)-N-propylpropanamide
N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-benzothiazole-5-carboxamide
{3-[(4-fluorophenyl)methyl]-1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}methanol
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methylpyrimidin-2-amine
2-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenoxy]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-cyclohexanecarbonyl-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(2-methylphenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
2-[(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)methyl]benzoic acid
N-[(2R,3R)-1'-[(3-ethoxy-4-methoxyphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
(4aR,7aS)-1-benzyl-4-(1-methyl-1H-pyrazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 4-[2-(4-fluorophenyl)piperidin-1-yl]butanoate
3-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-1-(2-methoxyacetyl)piperidine-4-carboxamide
6-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-ethyl-N-methylpyridin-2-amine
1-(pyridin-2-yl)-4-{[3-({1-[2-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}piperazine
6-(3-chlorothiophene-2-carbonyl)-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
N,3-dimethyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydroquinazoline-7-carboxamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-{3-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
1-(7,7-dimethyl-5-{[5-(propan-2-yl)pyrimidin-4-yl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
N-(oxan-4-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-(3,4-dimethylphenoxymethyl)-N-{[4-(morpholin-4-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
4-methyl-2-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
2-[5-chloro-2-(propan-2-yloxy)phenyl]-2-[4-(cyclopropylmethyl)piperazin-1-yl]acetic acid
6-({[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}methyl)-1,4-oxazepan-6-ol
N-[2-(dimethylamino)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)-N-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}acetamide
N-[2-(benzylsulfanyl)ethyl]-2-(methylamino)pyridine-4-carboxamide