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N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,5-dimethyl-1H-pyrazole
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-1,3-thiazole-5-carboxamide
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{1-[2-(2,5-dimethylphenyl)ethyl]piperidin-4-yl}ethan-1-ol
ethyl 4-(2-phenoxyethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxylate
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-hydroxy-4-(methylsulfanyl)butanamide
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2,4-difluoro-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
(3S,5S)-1-benzyl-N-(propan-2-yl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}propanamide
4-{2-methyl-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-2-yl}morpholine
1-methyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(cyclopropylmethyl)-2-(3-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-methoxyethyl)-N-methylacetamide
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
[(5-chloro-2,3-dimethoxyphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
6-(3-acetylphenyl)-3,4-dihydroquinazolin-4-one
1-(2-aminoethyl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-1H-1,2,3-triazole-4-carboxamide
N-(1-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-N,2-dimethylfuran-3-carboxamide
4-(9H-purin-6-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-pyrrol-1-yl)-1,3-thiazole
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-{[2-(pyridin-2-yl)-1H-imidazol-1-yl]methyl}-3-(thiophen-2-yl)propan-1-ol
4-{4-[3-(4-fluorophenoxy)piperidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}pyridine
1-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-{2-methylimidazo[1,2-a]pyridin-5-yl}urea
(3S)-4-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-[(5-ethylpyridin-2-yl)methyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-(2-ethylpiperidin-1-yl)propan-1-one
4-(4-acetylphenyl)-3-(4-hydroxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(1-benzothiophen-2-yl)-1H-pyrazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
1-(6-methyl-3-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}quinolin-2-yl)piperidin-3-ol
1-(4-{3-[(3,4-dimethoxyphenyl)amino]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
N-butyl-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
1-methyl-2-{[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
1-(3,5-dimethylphenyl)-3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}urea
N-ethyl-2-(4-{2-[2-(trifluoromethyl)phenyl]acetyl}piperazin-1-yl)acetamide
1-{[1-(2-methoxyphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
2-methoxy-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
N,N-dimethyl-2-({[(2-phenylethyl)carbamoyl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
methyl[(5-methylfuran-2-yl)methyl]{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
4-(3-{[1-(3-ethynylbenzoyl)piperidin-4-yl]oxy}benzoyl)morpholine
2-{[(6-methyl-2-propylpyrimidin-4-yl)amino]methyl}-3,4-dihydroquinazolin-4-one
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
7-cyclohexyl-2-(2-hydroxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
2-[(3S,4R)-3-cyclopropyl-4-acetamidopyrrolidin-1-yl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
2-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}-N-(oxolan-2-ylmethyl)benzamide
N-(2-methylpropyl)-5-{1-[2-(piperidin-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2,7-dioxo-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,3-diazepane-4-carboxamide