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({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methylpentanamide
2-(2-methoxyethoxy)-1-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
1-cyclohexyl-6-(pyridin-3-ylmethoxy)-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1,4-diazepan-2-one
3-[4-(2-methoxyethoxy)piperidin-1-yl]-5-(2-methylphenyl)-1,2,4-triazine
6-fluoro-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(2-fluorophenyl)-1-methyl-3-{2-[3-(3-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]({[6-(trifluoromethyl)pyridin-3-yl]methyl})amine
N-(2-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
5-(3-chlorobenzoyl)-N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 3-[(3S,4R)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
[5-(4-phenylazepane-1-carbonyl)furan-2-yl]methanol
6-ethyl-N-[1-(4-methanesulfonylphenyl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)pyridin-1-ium-1-olate
N-benzyl-5-{[4-(pyrimidin-4-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
(7S,8aS)-7-{2-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}-2-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-{4-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
3-(3-chlorophenyl)-4-methoxybenzamide
(4aS,7aR)-1-(1H-indole-2-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-9-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[(dimethylamino)methyl]phenyl}-N,N,5-trimethylpyrimidin-4-amine
2-(dimethylamino)-N-methyl-2-(4-methylphenyl)-N-(1,2-oxazol-3-ylmethyl)acetamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methyl-1-benzofuran-5-carbonyl)morpholine
N,N-dimethyl-3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decane-8-sulfonamide
2-(3-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}phenoxy)acetamide
8-methoxy-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[1-(3-phenylpropyl)-5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
2-{4-[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]piperidin-1-yl}acetamide
N-[(3R,4R)-3-hydroxy-1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-4-yl]pyridine-2-carboxamide
(2R,3R)-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-methoxy-1-[(4-methoxyphenyl)methyl]-4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1,4-diazepan-2-one
N-[(3S,4R)-1-(3-cyanopyridin-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
2-[4-(1-benzothiophene-2-sulfonamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
methyl 4-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]carbamoyl}amino)-3-methylbenzoate
7-[2-(benzyloxy)ethyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylate
2-[(4aR,7aS)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(pyridazine-3-carbonyl)pyrrolidin-3-yl]methanol
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-(pyridin-4-yl)propan-1-one
6-oxo-N-({1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)-1,6-dihydropyridine-3-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(9H-purin-6-yl)piperidin-4-amine
1-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methylpiperidin-2-one
6-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-tert-butyl-5-oxo-N-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrrolidine-3-carboxamide
2-(4-methoxyphenyl)-N-{[8-(pyridin-3-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
N-(1-{2-oxo-2-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
5-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione