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N-methyl-N-[2-(4-methylphenoxy)ethyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-[(4,6-dimethylpyrimidin-2-yl)methyl]-1λ6-thiane-1,1-dione
8-(1H-indol-3-ylmethyl)-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-2-(4-methylpiperazin-1-yl)aniline
(3aR,6aR)-2-[(5-fluoro-2-methoxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-fluorophenyl)-N-({7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-6-methoxy-1-methyl-1H-indole
2-(1-benzyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
6-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
3-benzyl-N-[2-(furan-2-yl)ethyl]-1,2-oxazole-5-carboxamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(3-fluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
2-[(4aR,7aS)-4-[(3-fluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
7-methanesulfonyl-4-methyl-2-[4-(3-phenylpiperidin-1-yl)piperidin-1-yl]quinazoline
2-methyl-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-5-sulfamoylbenzamide
3-[(3R,4S)-1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
5-chloro-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyridin-2-amine
4-oxo-4-[3-oxo-4-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-1-yl]butanamide
1-(4-methoxyphenyl)-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
2-{2-[(butan-2-yl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
6-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
(4S)-4-acetamido-5-oxo-5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pentanamide
2-{1-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)benzamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
(3S,4S)-1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
N-(3-methylbutan-2-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
ethyl 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]-4-(2-oxopyrrolidin-1-yl)benzamide
N-[4-(4-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}piperidin-1-yl)phenyl]cyclopentanecarboxamide
methyl 1-(3-methylbutoxy)-2-oxo-8-(3-phenylbutyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)oxan-4-amine
N-cyclopropyl-3-(1-methylpiperidin-4-yl)propanamide
2-[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
2-{3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
1-[2-(4-fluorophenyl)benzoyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-(pyridin-3-yl)propanamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}[(2-methoxyphenyl)methyl]amine
2-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-5-(dimethylamino)-2,3-dihydropyridazin-3-one
5-(2-chlorophenyl)-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methylfuran-2-carboxamide
1-methyl-5-[(2-methyl-1-benzothiophen-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
4-{1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-1λ6-thiane-1,1-dione
5-methyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
methyl (2S,4R)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-(dimethylamino)pyrrolidine-2-carboxylate
8-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
ethyl 4-(2-phenoxyethyl)-1-(phenylcarbamoyl)piperidine-4-carboxylate
3-(furan-2-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
2-hydroxy-N-(1H-imidazol-2-ylmethyl)-N-methyl-5-(1H-pyrrol-1-yl)benzamide