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N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-(3-ethoxypropyl)-2-[(3-methoxyphenyl)amino]butanamide
(3S,4R)-4-(2-methoxyphenyl)-1-(quinoline-7-carbonyl)pyrrolidine-3-carboxylic acid
2-(1H-imidazol-2-yl)-1-[3-methoxy-4-(pyrrolidin-1-yl)phenyl]-1H-imidazole
N-(1-ethyl-2-methyl-1H-indol-5-yl)-4-(5-methylpyrimidin-4-yl)piperidine-1-carboxamide
1-({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}amino)propan-2-ol
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(pyrimidin-2-yl)piperidin-3-yl]benzamide
2-(3-methyl-1,2,4-oxadiazol-5-yl)-1-(1,3-thiazol-4-ylmethyl)piperidine
2-(3-hydroxypiperidin-1-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-(2-methoxyphenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
(4aR,7aS)-1-ethyl-4-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-2-(1-ethylpiperidin-4-yl)-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
(4aS,8aR)-6-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-pyrazol-4-yl)butan-1-one
methyl(2-phenyl-1-{1-[3-(trifluoromethyl)benzoyl]piperidin-4-yl}ethyl)(pyridin-3-ylmethyl)amine
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)benzamide
1-[(3-fluorophenyl)methyl]-3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]urea
methyl 4-{[6-oxo-1-(2-phenylethyl)piperidin-3-yl]formamido}butanoate
5-[4-(4-methoxybutyl)piperazine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
(2E)-3-(2-chlorophenyl)-N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)prop-2-enamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
3-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
8-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
4-({2-[1-(1,3-thiazol-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-(4-chloro-1H-pyrazol-1-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
4-[2-(4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)propyl]-2-methoxyphenol
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-(2-ethyl-1H-imidazol-1-yl)propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3-chlorophenyl)methyl]piperidin-3-ol
13-(2,3-dimethoxyphenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
4-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
3-ethyl-4-{3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanoyl}piperazin-2-one
2-{2-[3-(morpholin-4-yl)azetidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
(1R,3s,6r,8S)-4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
1-phenyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-[carbamoyl(methyl)amino]-N-[(3R,4S)-1-(4-methylpent-3-en-1-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-[5-(2-methylbenzoyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}morpholine
N-[(2-fluorophenyl)methyl]-N-propyl-3-(1H-pyrazol-1-ylmethyl)benzamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1H-indole-5-carboxamide
3-cyclopropyl-5-(5-cyclopropyl-1,3-oxazol-4-yl)-1-(2-methoxyphenyl)-1H-1,2,4-triazole
N-ethyl-N-(2-hydroxyethyl)-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
5-{1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}-2-methoxyphenol
2-methoxy-N-({7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
1-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
5-methyl-14-[5-(2-methylpropyl)thiophen-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
6-[({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)amino]pyrazine-2-carboxamide
[(3aS,6aS)-2-{1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]piperidin-4-yl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol