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2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[2-methyl-2-(morpholin-4-yl)propyl]pyridin-2-amine
3-(4-benzyl-1H-pyrazol-5-yl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-(thiophen-3-yl)propan-1-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(morpholine-4-carbonyl)piperidin-1-yl]ethan-1-one
7-(1-ethyl-1H-pyrazole-3-carbonyl)-N,N-dimethyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-methyl-5-[5-(1H-1,2,4-triazol-1-ylmethyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
6-[2-butyl-4-(4-chlorophenyl)-5-oxopiperazine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
4-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]-1-(3-methoxyphenyl)piperazin-2-one
ethyl 4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine-1-carboxylate
4-(3-acetylphenoxy)-1-(cyclohexylmethyl)piperidine-4-carboxylic acid
ethyl 1-[7-oxo-2-(thiophene-3-amido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carbonyl]piperidine-4-carboxylate
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methoxyphenyl)methyl]acetamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(pyridin-4-yl)piperazin-1-yl]ethan-1-one
3-({[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
3-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenol
methyl 4-[(1-cycloheptylpiperidin-3-yl)carbamoyl]butanoate
methyl 5-{[(2,5-dimethylphenyl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-hydroxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)acetamide
N-[3-(1H-indol-2-yl)phenyl]-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
(3R)-N-({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)oxolan-3-amine
(2S,4S)-4-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-amido]pyrrolidine-2-carboxylic acid
1-[(2-fluorophenyl)methyl]-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-2-one
(1S,5R)-3-benzyl-6-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
3-(2,5-dimethylbenzoyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[2-hydroxy-3-(4-methoxy-2-{[(3,3,5,5-tetramethylcyclohexyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
4-(naphthalene-2-sulfonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1-{2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}pyrrolidin-2-one
6-ethoxy-4-methyl-2-{4-[(2,4,5-trimethoxyphenyl)methyl]-1,4-diazepan-1-yl}quinazoline
2-amino-4-(4-hydroxy-3-methoxyphenyl)-6-(5-methylthiophen-2-yl)pyridine-3-carbonitrile
1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
N-[(3,4-dimethoxyphenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methylpyrrolidine-2-carboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethyloxane-4-carboxamide
N-[(2R,3R)-1'-[(4-fluorophenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(furan-2-carbonyl)piperidine
1-(4-chlorophenyl)-5-methyl-4-[2-(3-methylphenyl)acetyl]piperazin-2-one
1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]azetidin-3-ol
1-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
methyl 3-[(3,5-dimethoxyphenyl)methyl]-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(pyridin-3-ylmethyl)azepan-4-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
1-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
6-fluoro-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N-(pyridin-4-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-1,2,3-triazole-5-carboxamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-{2-oxo-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}piperidine-4-carboxamide
2-[5-(4-cyano-1-methyl-1H-pyrrol-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid