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2-methyl-1-[(3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-pyrazol-5-yl)methyl]-1H-1,3-benzodiazole
2-{[(4-{[2-(2-methoxyphenyl)ethyl]amino}quinazolin-2-yl)methyl](propan-2-yl)amino}ethan-1-ol
N-[4-(furan-2-yl)phenyl]-3-(methanesulfonylmethyl)piperidine-1-carboxamide
3-(2-methylpropyl)-2-oxo-1-{1-[(pyridin-2-yl)carbamoyl]ethyl}-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
3-(4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}(1-phenylethyl)amine
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-N-ethylpyrimidin-2-amine
2-methyl-4-[4-({2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)phenyl]butan-2-ol
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(4-methylphenyl)methyl]acetamide
4-{5-[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridine
4-chloro-1-(pyrimidin-5-yl)-1H-indazole
5-(3-fluorophenyl)-N-[(4-phenyloxan-4-yl)methyl]-1,2,4-triazin-3-amine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
5-methoxy-2-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)pyridin-4-ol
4-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
1-(4-{4-[(prop-2-en-1-yl)amino]piperidin-1-yl}benzoyl)piperidin-3-ol
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[6-(methoxymethyl)pyrimidin-4-yl]pyrrolidin-3-yl]methanol
N-cyclopentyl-2-methyl-6-(piperidin-4-yl)-N-(prop-2-en-1-yl)pyrimidin-4-amine
3-(2-methoxyphenyl)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}propan-1-one
N-[(3,4-dimethoxyphenyl)methyl]-3-(2-oxoimidazolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
5-{1-[2-(4-chloro-2-methylphenoxy)propanoyl]piperidin-4-yl}-5-[(2-fluorophenyl)methyl]imidazolidine-2,4-dione
5-phenyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-{[4-(thiomorpholine-4-carbonyl)-1,3-oxazol-2-yl]methoxy}isoquinoline
1-cyclopentyl-N3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
2-{4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1H-pyrazol-1-yl}acetic acid
2-[1-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
10-methoxy-5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-[(1-benzyl-1H-imidazol-5-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(diphenylmethyl)-5-(ethanesulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[4-(3-methylphenyl)phenyl]-1-(oxolan-3-ylmethyl)piperidine-4-carboxamide
2-methyl-6-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]pyrimidin-2-amine
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(4-phenylbutanoyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(2-methoxyethyl)-2-[3-(4-methoxyphenyl)-1-(3-methylbutyl)-2,5-dioxopyrrolidin-3-yl]-N-(propan-2-yl)acetamide
5-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-[(3,4-dimethoxyphenyl)methyl]-6-(thiomorpholine-4-carbonyl)-1,3-benzoxazole
1-{2-[2-(4-methoxyphenoxy)acetamido]ethyl}-N-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
2-(dimethylamino)-N-{3-methyl-1-[7-(naphthalene-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
3-{4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}butan-1-ol
N-cyclopropyl-2-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methoxy)benzamide
(1R,3S)-N-(3,4-dichlorophenyl)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-4-ethenyl-N-methylbenzamide
5-ethyl-N-[1-(pyridin-4-yl)propan-2-yl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-{[3-methyl-7-(naphthalene-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(piperidin-1-yl)acetamide
methyl 2-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxylate
6-[(2-fluorophenyl)methoxy]-4-(furan-3-carbonyl)-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one