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4-[(6-methoxypyrimidin-4-yl)amino]-1-(propan-2-yl)pyrrolidin-2-one
6-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-N,N-dimethylpyrazine-2-carboxamide
4-[6-(methoxymethyl)pyridine-2-carbonyl]thiomorpholine
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
(2S,4R)-4-amino-N-methyl-1-{[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}pyrrolidine-2-carboxamide
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2-methoxyphenyl)ethan-1-one
N-{[7-(2,3-dimethoxybenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
2-[(1S,5R)-3-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[2-(diethylamino)ethyl]-N-ethyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 3-benzyl-1-(1H-pyrazole-4-carbonyl)piperidine-3-carboxylate
(4aS,7aR)-1-(3-methylfuran-2-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-methoxybenzamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(5-methylpyrazin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-fluorophenyl)-N-{2-[7-(1H-indol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
3-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
N-[3-(phenylsulfanyl)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyrrolidine-1-carboxamide
4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(2,4-difluorophenyl)methyl]-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
4-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]-1,3-dimethylpiperazin-2-one
N-benzyl-N-(cyclopropylmethyl)-2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}acetamide
2-{4-[(6-chloro-2H-chromen-3-yl)methyl]-1-cyclopentylpiperazin-2-yl}ethan-1-ol
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(3-fluorophenyl)-N-[(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
N-ethyl-6-[(1-phenylethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
5-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)pyridin-2-amine
benzyl(methyl)[(3-methylpyridin-4-yl)methyl]amine
1-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[(4-fluorophenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N2,N4,N4,5-tetramethyl-N2-(oxolan-2-ylmethyl)pyrimidine-2,4-diamine
methyl 7-oxo-9-[2-(piperidin-1-yl)ethoxy]-3-(quinolin-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[(3-fluorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3,4-difluorophenyl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
2-(dimethylamino)-2-(3-methylphenyl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
2-[3-(1H-imidazol-2-yl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(1H-imidazol-1-ylmethyl)piperidine
methyl 3-(cyclobutylmethoxy)-5-(dimethylcarbamoyl)benzoate
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(prop-2-en-1-yl)acetamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-1-ethyl-1H-pyrazole-3-carboxamide
1-[(1R,5S,6R)-6-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-3-azabicyclo[3.1.0]hexan-3-yl]-2-phenoxyethan-1-one
9-(dimethyl-1,2-oxazole-4-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
7-(cyclohexylmethyl)-2-(1H-imidazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-fluoro-N-({7-[4-(thiophen-2-yl)butanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
4-[1-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]thiomorpholine
N-cyclopropyl-5-methoxy-4-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-2-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-{2-[(2,6-dimethylphenyl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-3-methoxypropan-1-one
3-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)-N-(1,3-thiazol-2-yl)propanamide
2-[(1R,3S,3aS,6aR)-1-(hydroxymethyl)-5-methyl-3-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
5-({[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}methyl)-N,N-dimethylpyridin-2-amine