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2-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)imidazo[1,2-a]pyrimidine-2-carboxamide
ethyl 1-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidine-3-carboxylate
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4-(morpholine-4-carbonyl)pyridin-2-amine
5-(phenoxymethyl)-3-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-pyrazole
3-[3-(2-methoxyphenoxy)azetidin-1-yl]-5-phenyl-1,2,4-oxadiazole
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-methyl-3-{[(5-methylthiophen-2-yl)methyl]amino}-N-(oxan-2-ylmethyl)benzamide
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2,3-dihydro-1,4-benzodioxine-2-carboxamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-2-yl)ethan-1-one
ethyl[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amine
2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethan-1-one
8-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-5-(phenoxymethyl)-N-(pyrazin-2-ylmethyl)-1H-pyrazole-3-carboxamide
8-(2,1,3-benzoxadiazol-4-ylmethyl)-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
5-(dimethylamino)-2-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
N-({8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
6-methoxy-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidin-4-amine
4-{1-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-1-oxopropan-2-yl}-1,2-dihydrophthalazin-1-one
1-(1-{6-[(1,3-dihydroxypropan-2-yl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
3-(2,6-dimethylpyridin-3-yl)-1-{3-[(5-methylpyridin-2-yl)amino]propyl}urea
N-(3-hydroxypropyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1S,5R)-6-(1-benzofuran-2-ylmethyl)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-methoxy-5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]methanesulfonamide
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-4-(2-methylpropyl)benzamide
N-[3-(pyridin-4-yl)propyl]-6-[4-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
(1R,2R)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-phenylcyclopropane-1-carboxamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
9-methoxy-4-[(5-methylfuran-2-yl)methyl]-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-ethyl-N-methyl-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]pyrimidin-4-amine
N-[(1S)-2-hydroxy-1-phenylethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-{1-[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}furan-2-carboxamide
methyl 3-(2-acetylbenzoyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[2-methyl-3-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amino}methyl)-1H-indol-1-yl]acetamide
2-(3-methoxyphenyl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-(thiophene-2-carbonyl)-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-ethyl-4-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1,3-thiazole-5-carboxamide
(5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}furan-2-yl)methanol
N-{[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]methyl}-2-(4-methoxyphenyl)acetamide
1-(3-fluoro-2-methoxybenzoyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
(1R,5S,6S)-6-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
5-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-(5-{[3-(ethylcarbamoyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(4-ethylpiperazin-1-yl)-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
N-[(2-aminopyrimidin-5-yl)methyl]-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-{2-[4-(3-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-methoxy-N-[4-methyl-3-({methyl[2-(pyridin-2-yl)ethyl]carbamoyl}amino)phenyl]acetamide
4-(1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-3-yl)benzoic acid