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4-(3-hydroxy-3-methylbutyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
6-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[3-(methylsulfanyl)propyl]acetamide
2-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxy-N-methyl-N-propylpyrimidine-5-carboxamide
5-(2-methoxyethyl)-3-{[4-phenyl-5-(1-phenylethyl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
6-{3-[4-(2-chlorophenoxy)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(ethyl)(oxan-2-ylmethyl)amine
N-(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
{3-[(3-methoxyphenyl)methyl]-1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl}methanol
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
1-methyl-N-[3-(thiomorpholine-4-carbonyl)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-phenyl-2-(pyridin-4-yl)-4-[1-(thiolan-3-yl)piperidin-3-yl]pyrimidine
1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-4-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
3-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
6-methoxy-N-[(1R)-1-(3-methoxyphenyl)ethyl]pyrimidin-4-amine
methyl 2-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxylate
6-ethoxy-2-(thiomorpholin-4-ylmethyl)quinoline
3-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-benzyl-1-cyclopentyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(3-chloro-4-fluorophenoxy)-1-[3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
3-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
2-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-cyclopentyl-4-[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]-1,4-diazepane
ethyl 5-[(3-methylquinoxalin-2-yl)methyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[1-(3-methylbutyl)-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl]ethan-1-ol
2,2-dimethyl-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]thiomorpholin-3-one
5-methyl-N-(3-{5-methyl-4-[(3-methylbutanamido)methyl]-1,3-oxazol-2-yl}phenyl)thiophene-2-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-[(3,4-difluorophenyl)methyl]piperidin-3-amine
(1S,5R)-3-(2-amino-6-methoxypyrimidin-4-yl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-hydroxy-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-4-(thiophen-2-yl)butanamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-2-[3-(4-methoxyphenyl)-1-(3-methylbutyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]quinoline-2-carboxamide
1-{9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one
3-[2-(2-methoxypyrimidin-5-yl)-1H-imidazol-1-yl]quinoline
4-(4-fluorophenyl)-N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)-4-oxobutanamide
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2,6-dimethylquinoline-4-carboxamide
(3S,4S)-1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
2-(3-chlorophenoxy)-N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}thiomorpholine
4-(4-benzyl-1H-pyrazol-5-yl)-1-(1H-imidazol-2-ylmethyl)piperidine
1-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-cyclopentyl-4-[5-(ethanesulfonyl)thiophen-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(cyclobutylmethyl)-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
methyl 5-{[(2-chloro-6-fluorophenyl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(4-fluorophenyl)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-ol