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(1R,7S)-N-(furan-3-ylmethyl)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{3-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}-3-(4-ethylpiperazin-1-yl)propan-2-ol
2-methoxy-N-({8-[(2-methoxynaphthalen-1-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(morpholin-2-yl)acetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-phenylcyclopropan-1-amine
3-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-3-(4-methoxyphenyl)-1-(3-methylbutyl)pyrrolidine-2,5-dione
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)propanamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
6-[(2-chloro-3,4-dimethoxyphenyl)methyl]-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(prop-2-en-1-yl)-9-(quinoxalin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}azepan-2-one
7-(3,6-dimethylpyrazin-2-yl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-oxo-N-(2-phenoxyethyl)-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-(2,2-dimethyloxan-4-yl)-1-(6-methoxy-4-methylquinazolin-2-yl)piperidin-4-amine
(2S,4R)-4-amino-1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-N-ethylpyrrolidine-2-carboxamide
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-propyl-1,4-diazepan-6-yl]oxy}acetamide
4-hydroxy-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
4-(4-fluorophenyl)-1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}butan-1-one
4-[(2S,4R)-1-[(2-fluorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[(4-methoxyphenyl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)azepane-2-carboxamide
8-(2,3-dihydroxypropyl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-(naphthalen-2-ylmethyl)-N5-(2-phenoxyethyl)piperidine-3,5-dicarboxamide
N-(2-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
N-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
3-(3-methoxyphenoxymethyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
(2R,6R)-4-(4-fluorobenzoyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-(2-phenylethyl)piperidin-2-one
2-methoxy-N-[(2R,3R)-1'-[2-(methylsulfanyl)benzoyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-[1-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
1-(2-{1-[4-methyl-6-(methylsulfanyl)quinolin-2-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methylphenyl)methyl]acetamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-[3-(pyridin-3-yl)propyl]propanamide
1-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylbenzamide
7-fluoro-3-({[3-(4-fluorophenoxy)propyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
8-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}-2,8-diazaspiro[4.5]decan-3-one
(3R,4R)-4-cyclobutyl-3-methyl-1-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-4-ol
5-ethyl-2-{4-[(4-methylphenyl)methyl]piperazin-1-yl}pyrimidine
3-(1,4-diazepane-1-carbonyl)-N-[2-(1H-imidazol-4-yl)ethyl]benzene-1-sulfonamide
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-(3-phenylpropyl)pyrrolidin-2-one
N-[(3S,4R)-1-cyclopentanecarbonyl-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
8-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
dimethyl(2-{2-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-ethyl-N-[(4-methoxyphenyl)methyl]-2-methyl-N-propyl-1,3-thiazole-5-carboxamide