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(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
3-(4-hydroxyphenyl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
1-ethyl-N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[2-(cyclopent-1-ene-1-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-6-methylpyridine
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
5-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
(1R,9aR)-1-[({[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
6-ethyl-1,5-dimethyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
N-[2-(methylsulfanyl)ethyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
2-(adamantan-1-yl)-4-hydroxy-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]pyrimidine-5-carboxamide
(2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-{[(1r,4r)-4-hydroxycyclohexyl]carbamoyl}pyrrolidine-2-carboxylic acid
(2S,4R)-1-[(2-ethoxyphenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(2-fluorophenyl)methyl]-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
6-(2-aminoethyl)-2-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrimidin-4-amine
3-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(5-methylpyrazin-2-yl)methyl]urea
1-[3-(4-{[(adamantan-1-yl)amino]methyl}-2-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-2,3,6-trimethylquinoline
N-{[1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]methyl}-3-methylpyridine-2-carboxamide
3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-methoxybenzene-1-sulfonamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(morpholine-2-carbonyl)-1,4-diazepane
7-[3-(dimethylamino)phenyl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
4-[5-(propan-2-yl)thiophene-3-carbonyl]piperazine-2-carboxylic acid
1-(2-methoxyethyl)-6-oxo-N-{[4-(trifluoromethoxy)phenyl]methyl}piperidine-3-carboxamide
N-(3-fluoro-2-methylphenyl)-2-{[2-(pyridin-2-yl)ethyl]amino}acetamide
N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}thiomorpholine-4-carboxamide
5-cyclopropyl-N-[(3,5-dimethoxyphenyl)methyl]-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(thiophen-3-yl)acetamide
ethyl 1-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carboxylate
(4aS,7aR)-1-(2,5-dimethylfuran-3-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1,2,3,4-tetrahydroisoquinoline
8-[5-(trifluoromethyl)pyridin-2-yl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
3-[1-(pent-4-enoyl)piperidin-4-yl]-N-phenylpropanamide
[(3R,4R)-1-(1-benzylpiperidin-4-yl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-{6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}-5-fluoro-1H-1,3-benzodiazole
N-(1-methoxypropan-2-yl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-methoxy-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyridine-4-carboxamide
2-methyl-2-[2-(4-methylpiperazin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]propanoic acid
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[3-(pyridin-4-yl)-1H-pyrazol-1-yl]acetamide
N-(2-methoxyethyl)-N-methyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-{3-[(2,6-dichlorophenyl)methyl]-5-[(dimethylamino)methyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-ethyl-N-(oxolan-2-ylmethyl)acetamide
3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1-[1-(thiophen-2-ylmethyl)piperidin-3-yl]urea
7-cyclopropanecarbonyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
5-(4-acetyl-2-methoxyphenoxymethyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide