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2-[(2-methyl-1,3-oxazol-4-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
1-(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)propan-1-ol
2-(2-oxoazepan-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
methyl 3-{methyl[1-(2-phenylethyl)piperidin-3-yl]carbamoyl}propanoate
ethyl 1-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
({5-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[2-(azepan-1-yl)-2-phenylethyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
3-{1-[1-(3-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]piperidin-4-amine
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3,3-dimethylbutanamide
(2S)-N-(4-phenyl-1,2,3-thiadiazol-5-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
N-benzyl-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-(4-{[(5-methyl-1,2-oxazol-3-yl)methyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(4-chlorophenoxy)ethyl]-N-ethyl-2-methylimidazo[1,2-a]pyridine-6-carboxamide
(1S,5R)-6-benzyl-3-[(2,6-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-5-methoxy-3-methyl-1H-indole
(2S,4S)-4-amino-1-[2-(azocan-1-yl)acetyl]-N-ethylpyrrolidine-2-carboxamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]cyclobutanecarboxamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(6-methylpyridin-2-yl)methyl]piperidin-3-amine
4-(furan-2-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-2-(methoxymethyl)piperidine
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
4-[(4-ethynylphenyl)methyl]-9-(furan-2-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
N-(2-methoxyethyl)-5-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
ethyl 5-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-(1-ethyl-1H-pyrazol-4-yl)-1-(2-phenoxyethyl)-1H-1,2,3-triazole
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2,3-dihydro-1H-inden-2-amine
methyl 8-(2-benzyl-1,3-thiazole-4-carbonyl)-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-amino-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-propoxybenzamide
1-[(2-methoxyphenyl)methyl]-3-(1,3,4-thiadiazol-2-yl)urea
1-(4-fluorobenzenesulfonyl)-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrrolidine
4-(1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
1-[(2R)-oxolane-2-carbonyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
(3R,4R)-1-[(2-methoxynaphthalen-1-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
2-{[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-6-methylquinolin-4-ol
1-acetyl-N-[4-(3-fluorophenyl)phenyl]pyrrolidine-2-carboxamide
N-{1-[7-(cyclohexylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-methylbenzamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-(1-phenylpiperidin-4-yl)acetamide
6-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-2-(3-methylphenyl)-3,4-dihydropyrimidin-4-one
2-methoxy-1-(1'-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
3-(2-methoxyphenyl)-5-[1-(1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazole
8-(4-cyclopentylpyrimidin-2-yl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one