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6-({4-[methyl(phenyl)amino]phenyl}methyl)-N-(pyridin-3-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-cyclopropyl-6-methyl-2-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
(2S,4R)-1-{[4-(benzyloxy)phenyl]methyl}-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
(3S,7S)-5-[2-(methylsulfanyl)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
4-[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N-(propan-2-yl)pyridine-2-carboxamide
5-{3-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
6-(cyclopropylmethoxy)-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
methyl 3-{4-[(3-benzoylpiperidin-1-yl)methyl]-1H-pyrazol-1-yl}propanoate
1-{5-[(6-ethyl-2-methylpyrimidin-4-yl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
(1-{[2-(benzyloxy)phenyl]methyl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol
N-({1-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidin-3-yl}methyl)cyclopropanecarboxamide
9-(5-ethylfuran-2-yl)-4-methyl-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
N-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]thian-4-amine
(3R,4R)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-(1H-imidazol-4-ylmethyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
N-benzyl({4-[2-(pyridin-2-yl)ethyl]phenyl}amino)sulfonamide
N-[4-(furan-2-yl)butan-2-yl]-3-azaspiro[5.5]undecan-9-amine
2-(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-thiazole
(1R,3S,4S)-N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-hydroxy-4,7,7-trimethylbicyclo[2.2.1]heptane-1-carboxamide
2-[4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
N-[(3S,4R)-1-(4-cyclopentylpyrimidin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-3-(thiophene-2-carbonyl)piperidine
N'-(4-methylphenyl)-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}propanediamide
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-5-(1H-imidazol-1-ylmethyl)pyridine
3-(2-chlorophenyl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)propanamide
N-ethyl-5-(1H-indol-1-ylmethyl)-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-3-carboxamide
N-(oxan-2-ylmethyl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
4-[(3,3-dimethyl-4-phenylpyrrolidin-1-yl)sulfonyl]morpholine
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxy-2-methylpropanamide
2-[methyl({4-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl})amino]ethan-1-ol
N-(2-{1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}ethyl)acetamide
2-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
methyl 5-{[(2-chlorophenyl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[1-(propan-2-yl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
8-{[(2-fluorophenyl)methyl]carbamoyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1-[4-(pyrrolidin-1-yl)butyl]-1H-imidazole
(2S)-3-(4-hydroxyphenyl)-2-[2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamido]propanamide
N-(2,4-dimethoxyphenyl)-3-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]propanamide
N-(propan-2-yl)-2-[4-(2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetyl)piperazin-1-yl]acetamide
1-[2-(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
N-({7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-(4-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)acetamide
5-butyl-1-(4-chlorophenyl)-4-[2-(2-methyl-1H-imidazol-1-yl)acetyl]piperazin-2-one
[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
N-cyclopropyl-3-{1-[(3,5-difluorophenyl)methyl]piperidin-3-yl}propanamide
1-[(3,4-dimethoxyphenyl)methyl]-2-(1H-imidazol-2-yl)-1H-imidazole