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1-({4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}methyl)piperidine
(2S,3S)-2-amino-1-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-3-methylpentan-1-one
ethyl 1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxylate
5-ethyl-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,3,4-oxadiazol-2-amine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-(3-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
4-{[2-(difluoromethoxy)phenyl]methyl}-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
N-({8-cyclopropanecarbonyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(7-methyl-2-oxo-2H-chromen-4-yl)acetamide
6-{1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
3-(2-chlorophenyl)-1-(2-methoxyethyl)-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{[(5-methylfuran-2-yl)methyl]amino}pyridine-3-carboxamide
9-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
7-phenyl-2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-ethyl-5-{[(5-fluoro-2-methylphenyl)methyl]amino}-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 4-{[(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-2-(dimethylcarbamoyl)pyrrolidin-1-yl]methyl}benzoate
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
4-(5-chloro-3-phenyl-1H-indole-2-carbonyl)piperazin-2-one
1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-amine
4-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperazine-2-carboxylic acid
5-methyl-2-(2-methylquinolin-5-yl)pyrimidin-4-amine
1-({4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)-1H-1,3-benzodiazole
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(9H-fluoren-9-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[(4-methylphenyl)methyl]propanamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(morpholin-4-yl)acetamide
2-[2-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-[4-(1H-imidazol-1-yl)phenyl]-3-[1-(oxolan-2-ylmethyl)piperidin-4-yl]urea
5-(2-chlorophenyl)-N-[2-(pyridin-4-yl)ethyl]furan-2-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propan-2-ol
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
2-amino-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)pyridine-4-carboxamide
N-(1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-{1,3-dioxo-2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine-4-carboxamide
4-fluoro-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
N-[2-ethoxy-5-(trifluoromethyl)phenyl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
N-(1-benzylpyrrolidin-3-yl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
5,7-dimethyl-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
1-{4-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-1-yl}ethan-1-one
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-(pyridin-2-yl)piperazine
N-{3-[(methylcarbamoyl)methyl]phenyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
6-(4-chlorophenyl)-N-ethyl-N-(pyridin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-methylpyrimidine-5-carboxamide
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-methyl-1H-pyrazole-4-carboxamide
ethyl 4-[1-(4-oxo-3,4-dihydrophthalazine-1-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
6-{3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carbonitrile
2-(hydroxymethyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide