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2-methoxy-N-methyl-N-(pyrimidin-4-ylmethyl)quinoline-4-carboxamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanamide
N-[(2R,3R)-1'-(3,5-difluorobenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
(2-{2-[1-(8-methoxyquinolin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
[(3,5-dimethoxyphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
1-[benzyl(methyl)amino]-3-[4-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-(2-fluorophenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})(pyridin-3-ylmethyl)amine
N-(2-methyl-4-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]carbamoyl}phenyl)furan-2-carboxamide
1-{5-[(diethylamino)methyl]-2-phenylfuran-3-carbonyl}azepan-4-amine
ethyl(oxolan-2-ylmethyl){[1-(piperidin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl}amine
N-(adamantan-2-yl)-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
2-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2R,4R,6S)-2-(4-chlorophenyl)-6-[2-(ethylamino)pyrimidin-5-yl]oxan-4-yl]acetamide
8-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-amino-4-methyl-N-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}pyrimidine-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1H-1,2,3-triazole-5-carbonyl)piperazine
2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxo-N-(propan-2-yl)acetamide
6-[2-(3-chlorophenoxy)propanoyl]-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-{2-[4-(piperidin-1-yl)benzoyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
methyl 7-oxo-9-(propan-2-yloxy)-3-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(2H-1,3-benzodioxol-5-yl)-1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
6-ethyl-N,N-dimethyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
5-{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{[7-(2,4-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}benzenesulfonamide
2-[2-(5-benzyl-4-phenyl-1H-imidazol-1-yl)ethoxy]ethan-1-ol
9-[3-(5-methylfuran-2-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-[(diethylamino)methyl]-5-ethyl-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]furan-2-carboxamide
(1R,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(5-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(4aR,7aS)-1-ethyl-4-[(5-methoxy-1H-indazol-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(oxan-4-yl)piperidine
4-phenyl-1-[2-(1,3-thiazol-4-yl)acetyl]piperidine-4-carbonitrile
(3R,4R)-N-[(4-chlorophenyl)methyl]-3-hydroxy-3,4-dimethylpyrrolidine-1-carboxamide
6-(4-fluorophenyl)-N-(2-hydroxyethyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-({2-[(2-carbamoylethyl)(propan-2-yl)carbamoyl]phenyl}amino)acetic acid
N-[(2-{4-[5-(methoxymethyl)thiophene-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-methyl-5-{2-oxo-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorothiophene-2-carboxamide
1-[4-(2-phenoxyethyl)piperazin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-(cyclobutylmethyl)-3-hydroxy-3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
2-(5-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl)acetic acid
2-amino-4-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-6-(pyridin-2-yl)pyridine-3-carbonitrile
13-(3-chloro-5-fluoro-4-methoxyphenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
3-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-1,2-benzothiazole