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N-[2-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)ethyl]pyridine-4-carboxamide
1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}-3-[3-(pyridin-3-yl)propyl]urea
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
1-[(3-methoxyphenyl)methyl]-4-[(4-{[(5-methylfuran-2-yl)methyl]amino}quinazolin-2-yl)methyl]piperazin-2-one
5-(methoxymethyl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]thiophene-2-carboxamide
1,3,5-trimethyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1H-pyrazole-4-carboxamide
methyl 1-{3-[(2,3-difluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
1-[4-({4-[4-(pyrrolidin-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
ethyl 2-{1-[2-(1-cyclopentyl-3-oxopiperazin-2-yl)acetamido]cyclohexyl}acetate
1-cyclopentyl-N-{[1-(dimethylamino)cyclohexyl]methyl}-6-oxopiperidine-3-carboxamide
N-({5-[(2-butyl-1H-imidazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
(1R,2S,6R,7S)-4-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-4-azatricyclo[5.2.2.02,6]undecane
3-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-methylbenzoic acid
1-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[4-(5-methylfuran-2-yl)phenyl]methyl})(pyridin-4-ylmethyl)amine
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(methylsulfanyl)acetamide
2-(3,4-dichlorophenyl)-4-(2-methoxy-6-methylbenzoyl)morpholine
3-[(3-fluorophenyl)methyl]-N-(1-phenylcyclopropyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{3-[2-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-4-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
N-(3-phenylpropyl)-6-[4-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
N-[(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)methyl]quinoline-8-sulfonamide
3,5-dichloro-4-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]benzamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(thiophen-2-yl)acetamide
7-(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)-3-methyl-3,4-dihydroquinazolin-4-one
N-[2-(dimethylamino)-3-methylbutyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-chloro-5-({[2-(2-oxopiperidin-1-yl)ethyl]carbamoyl}amino)-N-propylbenzamide
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}urea
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)pyrazine-2-carboxamide
1-[2-chloro-5-(piperidine-1-carbonyl)phenyl]-3-(thiolan-3-yl)urea
1-{4-[2-(4-methylphenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
3-[5-(5-methoxypentyl)-1,2,4-oxadiazol-3-yl]pyridazine
1-[2-(2,3-dimethoxyphenyl)ethyl]-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
2-fluoro-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]benzamide
methyl (2S,4S)-1-[(4-methylphenyl)methyl]-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
2-(3-methoxypropyl)-8-[6-(propan-2-yl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(1H-imidazol-1-yl)ethyl]-3-{[(5-methyl-1H-pyrazol-3-yl)methyl]sulfamoyl}benzamide
3-(2-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-(pyridin-4-yl)propan-1-one
5-cyclobutanecarbonyl-1'-(oxane-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
9-methoxy-3-[(4-phenylphenyl)methyl]-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-[1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-1-oxopropan-2-yl]propanamide
methyl 3-[2-(2H-indazol-2-yl)acetyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-ethyl-4-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
6-methyl-1-(2-methylphenyl)-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-one
2-(morpholin-4-ylmethyl)-4-(pyridin-4-ylmethyl)-1,4-oxazepane
8-methyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]-4-(pyrrolidine-1-carbonyl)quinoline
5-{[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]sulfonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione