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4-(1-benzofuran-2-carbonyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
4-(1H-imidazole-4-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
(4aS,8aR)-6-[3-(1,2-oxazinan-2-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
(1S,5R)-3-(quinolin-4-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-butyl-4-[2-(pyridin-2-yl)acetyl]piperazin-2-one
1-benzyl-8-[(3-methoxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-cyclopentyl-2-[3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
6-methyl-4-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]quinoline
1-(2-{[4-(trifluoromethyl)pyrimidin-2-yl]amino}ethyl)imidazolidin-2-one
5-[(1-benzothiophen-2-ylmethyl)(methyl)amino]-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 4-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}benzoate
4-(benzyloxy)-N-methyl-N-(1,3-thiazol-2-ylmethyl)butanamide
ethyl 2-{1-[2-(2-fluorophenoxymethyl)-1,3-oxazol-4-yl]-N-methylformamido}acetate
1-[5-(1,3-dimethyl-1H-pyrazol-4-yl)-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
1-(cyclopropylmethyl)-N-ethyl-5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{4-[4-(2-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[2-(2-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(5-ethyl-1,3-oxazole-4-carbonyl)-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
(3S,9aR)-3-(propan-2-yl)-8-(pyridin-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-methoxy-9-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1-oxa-9-azaspiro[5.5]undecane
(3R,4R)-1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
2-methoxy-N-methyl-N-(quinolin-5-ylmethyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)acetamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-ethyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
4-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-1-cyclopentylpiperazin-2-one
(2S,4R)-N-[2-(dimethylamino)ethyl]-1-(9H-fluoren-2-ylmethyl)-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
methyl 3-(2-fluorobenzamido)-6-{[methyl(2-phenylethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]piperidin-3-amine
1-cyclobutanecarbonyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)piperidine-4-carboxamide
5-(2-methylphenyl)-4-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}-2-(pyridin-4-yl)pyrimidine
N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-(pyrimidin-2-yl)piperidin-4-amine
3-[1-(4-cyanopyridin-2-yl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[(3-hydroxypyrrolidin-3-yl)methyl]-1-(2-phenylethyl)piperazin-2-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclohexyl-N-methylacetamide
3-cyano-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
4,6-dimethyl-2-oxo-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-dihydropyridine-3-carboxamide
N-(1,2,3,4-tetrahydronaphthalen-1-yl)-3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzamide
1-{4-[4-(2-chlorophenoxy)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
6-(1-ethyl-1H-pyrazol-4-yl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
3-benzyl-4-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)piperazin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2,3-dihydro-1-benzofuran-7-carbonyl)piperidin-3-ol
(3R,5S)-N-[3-(dimethylamino)propyl]-1-[(4-hydroxyphenyl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
[(3,4-difluorophenyl)methyl]({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
1-{[(1-cycloheptylpiperidin-3-yl)carbamoyl]methyl}piperidine-4-carboxamide
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
6-(3-{[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-4-(2-oxopyrrolidin-1-yl)benzamide