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(2S)-2-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidine-1-carboxamide
dimethyl({[(1R,5S,6S)-3-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
9-[(2R)-2-amino-3-methoxypropanoyl]-2-(4-hydroxybutyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-methyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-ethyl-N-methyl-3-(propan-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
2-(4-{[4-(furan-2-yl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
N-cyclopropyl-3-[1-(quinolin-8-ylmethyl)piperidin-3-yl]propanamide
2-{4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
(5-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyrrolidin-3-ylmethyl)amine
5-cyclopentanecarbonyl-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-methyl-5-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1'-{2-methyl-2,8-diazaspiro[4.5]decane-3-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]
N-{3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}methanesulfonamide
(2S,4S)-1-methyl-4-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamido]pyrrolidine-2-carboxylic acid
N-[(3R,4S)-1-(3-hydroxypropyl)-4-propylpyrrolidin-3-yl]-2-(4-methyl-1H-pyrazol-1-yl)acetamide
N-[2-(4-hydroxyphenyl)ethyl]-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-ethyl-N-(2-hydroxyethyl)-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-(2,3-dihydro-1H-inden-2-yl)-2-hydroxy-4-(methylsulfanyl)butanamide
N,5-dimethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(4-{[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-ol
ethyl 1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
2-[(3aS,6aS)-1-[(3,5-difluorophenyl)methyl]-octahydropyrrolo[3,4-b]pyrrol-5-yl]-1,3-benzoxazole
2-(1-methyl-4-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}piperazin-2-yl)ethan-1-ol
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
2-[(4-methoxyphenyl)methyl]-4-[4-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-{5-[3-(pyrrolidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
1-methyl-2-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidine-1-carbonyl)-1H-indole
N-[(3S,4R)-1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1,3-dimethyl-2,6-dioxo-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
ethyl 1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazole-2-carboxylate
3-methoxy-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)propanamide
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-[2-(trifluoromethyl)morpholin-4-yl]propanamide
(1S,5R)-6-(5-chloro-2-methoxybenzenesulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
methyl (2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-[methyl(1,2-oxazol-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-4-(4H-1,2,4-triazol-4-yl)piperidine
9-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(1r,4r)-4-({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)cyclohexan-1-ol
1-[(4-fluorophenyl)methyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
methyl[(5-phenyl-1H-pyrazol-3-yl)methyl][(3-{[1-(pyridine-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
N-methyl-2-oxo-1-phenyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrrolidine-3-carboxamide
(5S,9aS,9bS)-5-(3,5-dimethoxyphenyl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(3-methoxyphenyl)methyl]-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
3,5-dimethoxy-N-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]methyl}benzamide
5-fluoro-N-methyl-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
4-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]piperazine-2-carboxylic acid
N,N-dimethyl-5-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-amine