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1-(2-methoxy-4-{1-oxa-7-azaspiro[3.5]nonan-7-ylmethyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
6,6-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5-oxothiomorpholine-3-carboxamide
3-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
(2-methylpropyl)(pyridin-2-ylmethyl){[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-cyclopropyl-5-oxo-N-[3-(pyridin-2-yl)propyl]pyrrolidine-3-carboxamide
2-(2-{[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenoxy)ethan-1-ol
3-[(3R,4S)-1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-4-(dimethylamino)piperidin-3-yl]propan-1-ol
ethyl 1-(furan-3-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
2-cyclopropyl-4-phenyl-9-(pyridazine-3-carbonyl)-2,9-diazaspiro[5.5]undecane
3-{4-[(2-hydroxyethyl)amino]quinazolin-6-yl}phenol
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
4,6-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
N-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-methyl-N-(2-phenylethyl)-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-[(2-fluorophenyl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
5-ethyl-2-{1-[2-methoxy-1-(pyridin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(piperidin-4-ylmethyl)benzamide
1-(2-chlorophenyl)-4-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperazin-2-one
2-[4-(1-cyano-1-methylethyl)phenyl]pyridine-4-carboxamide
4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-[3-(trifluoromethyl)benzoyl]piperidine
1-cyclopropyl-N-(piperidin-3-ylmethyl)-1H-pyrrole-2-carboxamide
N-{4-[1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]phenyl}-N-methylmethanesulfonamide
methyl[(5-phenyl-1,2-oxazol-3-yl)methyl](1,3-thiazol-2-ylmethyl)amine
4-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-{4-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-(cyclohexylmethyl)-N3-cyclopropyl-N5-ethyl-4-oxo-N3-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-[(1H-imidazol-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
1-[2-(dimethylamino)ethyl]-5-oxo-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]pyrrolidine-3-carboxamide
1-{3-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-3-oxopropyl}azepan-2-one
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]pyrazine-2-carboxamide
N-({1-[(1-methylpiperidin-4-yl)methyl]piperidin-4-yl}methyl)but-3-enamide
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-(2-phenoxyethyl)-1,2-oxazole-3-carboxamide
3-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
8-[(3,4-dimethoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-({[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)-1,2-dihydrophthalazin-1-one
1-(2-fluorobenzoyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[4-({methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenyl]acetamide
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-1-(oxan-4-yl)piperidine-3-carboxamide
N-{2-cyclobutyl-1-methyl-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-7-yl}oxolane-2-carboxamide
3-[(4-fluorophenyl)formamido]-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)propanamide
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
N2-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-methylpyrimidine-2,4-diamine
2-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-benzofuran-5-carboxamide
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-[4-(methylsulfanyl)benzoyl]piperidine
[1-(2-fluorobenzoyl)-3-[(2-fluorophenyl)methyl]piperidin-3-yl]methanol