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7-(3,6-dimethylpyrazin-2-yl)-4-(3-methoxypyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(1-methyl-1H-pyrazol-4-yl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]urea
2-(methylamino)-N-{[8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}pyrimidine-5-carboxamide
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methanol
4-{1-[2-(4-methoxyphenoxy)ethyl]piperidin-4-yl}pyridine
methyl N-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})carbamoyl]methyl}carbamate
8-[(3-ethoxy-2-hydroxyphenyl)methyl]-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2,6-dimethyl-8-({3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}amino)octan-2-ol
(2E)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2-methyl-N-(oxolan-2-ylmethyl)but-2-enamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
4-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1,4-dithiepan-6-amine
2-{[(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
(4aR,8aR)-2-methanesulfonyl-7-[(3-phenyl-1H-pyrazol-4-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
1'-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
ethyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl](pyridin-4-ylmethyl)amine
4-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-4H-1,2,4-triazole
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(6-ethylpyrimidin-4-yl)-N-methylpiperidin-3-amine
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
5-(3-acetylphenoxymethyl)-N-methyl-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-[(3-methoxyphenyl)methyl]-5-(morpholine-4-carbonyl)piperidin-2-one
4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-2-one
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(piperidin-1-yl)pentan-1-one
2-(4-fluorophenyl)-4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}morpholine
1-(5-chloro-2-methoxyphenyl)-5-(oxolan-3-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-(2,4-difluorophenyl)-2-[4-(1H-1,2,4-triazole-5-carbonyl)morpholin-3-yl]acetamide
4-(4-chlorophenoxy)-N-(2-methanesulfonylethyl)piperidine-4-carboxamide
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]pent-4-en-1-one
2-methyl-5-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrimidine
(1s,4s)-4-{4-[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
3-methyl-7-[2-(pyridin-2-yl)ethyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[3-(cyclohexylsulfanyl)propyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-6-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
4-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carbonyl)-6-methylpyrimidin-2-amine
3-(2,6-dimethoxypyridin-3-yl)-1-methyl-1-(oxan-2-ylmethyl)urea
1-{4-[(4-hydroxybutyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
6-fluoro-2-oxo-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2-dihydroquinoline-4-carboxamide
N-(pyridin-3-ylmethyl)-1-{1-[2-(pyridin-4-yl)acetyl]piperidin-4-yl}piperidine-4-carboxamide
3-(2-fluorophenyl)-N-{[8-(pyridine-2-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
1-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
6-[({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]pyrimidin-4-ol
(2S,4S)-4-amino-N,N-diethyl-1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidine-2-carboxamide
N-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]thiophene-2-carboxamide
2-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-4-methoxyphenol
3,5-dimethoxy-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-[(1S,2R)-2-aminocyclobutyl]-4-(1H-pyrazol-1-yl)benzene-1-sulfonamide
2-{5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrazol-3-yl}pyridine