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2,2-dimethyl-N-(1-{1-[(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
4-{4-[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]piperazin-1-yl}quinazoline
1-(3-chloro-2-fluorobenzoyl)-3-(3,4-dimethoxybenzoyl)piperidine
N-ethyl-5-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)pyrimidin-2-amine
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-5-methoxy-1-methyl-1H-indole-2-carboxamide
methyl 2-{[5-(4-fluorophenyl)-4-[1-(pyrazine-2-carbonyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3,3-dimethylbutanamide
5-[(methylsulfanyl)methyl]-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)furan-2-carboxamide
N-methyl-N-[(5-{[methyl(quinolin-5-ylmethyl)amino]methyl}furan-2-yl)methyl]methanesulfonamide
(3R)-1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}pyrrolidin-3-ol
1-(1,3-benzoxazol-2-yl)-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-amine
methyl 3-[(3-{[(2-fluorophenyl)methyl]carbamoyl}-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-yl)amino]propanoate
N-(2-{4-[(1-methyl-1H-indol-2-yl)methyl]morpholin-2-yl}ethyl)acetamide
3-[2-(furan-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]phenol
(4aS,7aR)-1-(furan-2-ylmethyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-{2-[1-(propan-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
(1S,5R)-1,3,3-trimethyl-N-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)-6-azabicyclo[3.2.1]octane-6-carboxamide
4-{1-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-1H-1,2,3-triazol-4-yl}benzoic acid
2-methoxy-1-(4-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
1-{2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
6-[(3-ethoxy-2-hydroxyphenyl)methyl]-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
5-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
1-[(2-fluorophenyl)methoxy]-8-(furan-3-ylmethyl)-1,8-diazaspiro[4.5]decan-2-one
7-fluoro-2-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}quinoline-4-carboxamide
3-methoxy-N-(2-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,2,3,4-tetrahydroisoquinolin-7-yl)propanamide
N-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
N-[(2R,3R)-1'-{[2-(furan-2-yl)phenyl]methyl}-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(6-methoxypyridin-3-yl)-1H-indazol-1-yl]acetamide
N-{3-[methyl(phenyl)amino]propyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-1,3-benzodiazole
ethyl 4-[(4-methoxyphenyl)methyl]-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine-4-carboxylate
N-[4-(2-fluorophenoxy)phenyl]-1-(pent-4-enoyl)piperidine-4-carboxamide
N-methyl-2-(2-methylfuran-3-amido)-N-[2-(4-methylphenoxy)ethyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-(2-{[(1,3-dimethylpyrrolidin-3-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
5-(2-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
methyl 3-(1-ethylpiperidine-3-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[2-(4-fluorophenyl)morpholin-4-yl]propan-1-ol
3-(3-chlorobenzoyl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
methyl 8-{[2-(difluoromethoxy)phenyl]methyl}-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
{3-[(3-methoxyphenyl)methyl]-1-[(3-methylquinoxalin-2-yl)methyl]piperidin-3-yl}methanol
(3S,4S)-4-(naphthalen-2-yl)-1-(9H-purin-6-yl)piperidin-3-ol
N-[4-(dimethylcarbamoyl)-2-methylphenyl]-4-(prop-2-en-1-yl)piperazine-1-carboxamide
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}acetamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
N-ethyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
N-[1-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide