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3-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-4H-chromen-4-one
N5-{[2-(furan-2-yl)phenyl]methyl}-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
N-[1-(1H-indol-5-yl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-4-(1H-pyrrol-1-yl)benzamide
1-methyl-4-[(4-methyl-5-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]piperazine
1-methyl-3-(2-methylpropyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
methyl 3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-methyl-2-oxo-N-[(3-phenylphenyl)methyl]-1,2-dihydropyridine-4-carboxamide
(1S,6R)-3-methyl-9-[2-(phenylamino)pyrimidine-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(ethylsulfanyl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
(2E)-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-phenylprop-2-en-1-one
8-methoxy-N-[(3-methylpyridin-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
N-(2-phenylethyl)-1-{1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-4-yl}piperidine-3-carboxamide
3-hydroxy-3-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}-1-(2-methoxyethyl)piperidin-2-one
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-3-(3-methoxyphenyl)propanamide
N-[2-(3-methoxyphenyl)-1-{1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}ethyl]-N-methylpyridine-2-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy]-N-methylacetamide
methyl N-{2-oxo-2-[9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]ethyl}carbamate
phenyl({1-[1-(thian-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl})methanol
N-{2-[2-(5-oxopyrrolidin-2-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-4-carboxamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-4-(2-oxopyrrolidin-1-yl)benzamide
5-(cyclohexylamino)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-(benzyloxy)-4-[(2-methyl-1H-imidazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-(4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
(1S,2S)-2-[4-phenyl-5-(quinolin-5-yl)-1H-imidazol-1-yl]cyclohexan-1-ol
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
(1S,5R)-3-{[4-(propan-2-yl)phenyl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2R,3R)-2-methoxy-1'-[3-(morpholin-4-yl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-(4-methoxyphenyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-[4-chloro-3-({[3-(4-methyl-1H-pyrazol-1-yl)propyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
N-cyclopropyl-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(naphthalen-2-yloxy)-1-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]propan-1-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]ethan-1-one
3-(but-2-yn-1-yl)-5-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
3-(1H-imidazol-1-ylmethyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
2-methyl-N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-[3-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-oxopropyl]acetamide
[(1-benzylpiperidin-4-yl)methyl]({[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-(furan-3-ylmethyl)-N-methyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[2-(2,4-dimethoxyphenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-6-(2-methoxyethyl)-3-{2-methylthieno[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 3-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]acetamide
2-methoxy-2-methyl-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-[4-(2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamido)phenyl]pentanamide
[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amine