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3-(1-butyl-1H-imidazol-2-yl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
2-oxo-8-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N2-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N2,N4,N4,5-tetramethylpyrimidine-2,4-diamine
4-[(4-methyl-5-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
1-cyclopropyl-N-[2-(2-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-(methylamino)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)pyridine-3-carboxamide
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
3-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-5-propyl-1-benzofuran-2-carboxamide
N,N-bis(prop-2-en-1-yl)-2-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)acetamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]benzamide
N-[(1-ethylpyrrolidin-3-yl)methyl]-N-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-fluoro-4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
4-fluoro-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]benzamide
N-[(3,4-dimethoxyphenyl)methyl]-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
7-(2-hydroxyethyl)-2-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[4-(4-cyclohexylpiperazine-1-carbonyl)piperidin-1-yl]-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-butyl-1-[(2-chlorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
6-(2,5-dimethylfuran-3-yl)-N-(2-hydroxyethyl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(3-methyl-1H-pyrazol-1-yl)-1-{4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
6-(2-chlorophenyl)-N-[2-(methylsulfanyl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-{5-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
methyl 1-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]piperidine-4-carboxylate
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
2-methoxy-5-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine
1-[(3S,4R)-1-[3-(4-fluorophenoxy)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
3-[(3R,4S)-1-[2-(4-ethylphenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-methyl-N-({3-methyl-7-[(2E)-4-methylpent-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-3-carboxamide
5-ethyl-N-methyl-N-(pyrimidin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-(isoquinolin-1-yl)phenol
4-(2-{1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}ethyl)phenol
(2S,4R)-1-benzyl-N-ethyl-4-{[(2-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-cyclohexyl-3-(2-fluorophenyl)-3-{2-oxo-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
8-(2,6-dimethylpyrimidine-4-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
1-(2-{1-[2-(1H-imidazol-5-yl)ethyl]-3-phenyl-1H-1,2,4-triazol-5-yl}ethyl)-4-methylpiperazine
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-phenylpropyl)piperidine
5-{3-[3-(2-chlorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
4-{1-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-imidazol-2-yl}benzamide
N-(2,3-dihydro-1H-inden-4-yl)-4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carboxamide
N4-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N-[3-methyl-1-(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]acetamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
methyl 1-[(3R,5S)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 6-(2-{[2-(3-methyl-1H-pyrazol-1-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]butan-1-one
2-phenoxy-N-({7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(1R,2R)-N-(1-methylpiperidin-4-yl)-2-phenyl-N-(2-phenylethyl)cyclopropane-1-carboxamide
5-[({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one